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Fragment-based covalent ligand screening enables rapid discovery of inhibitors for the RBR E3 ubiquitin ligase HOIP
Johansson, Henrik, Tsai, Yi-Chun Isabella, Fantom, Ken, Chung, Chun-Wa, Kümper, Sandra, Martino, Luigi, Thomas, Daniel A, Eberl, H Christian, Muelbaier, Marcel, House, David, Rittinger, KatrinLanguage:
english
Journal:
Journal of the American Chemical Society
DOI:
10.1021/jacs.8b13193
Date:
January, 2019
File:
PDF, 3.33 MB
english, 2019