Optimization of an azetidine series as inhibitors of colony stimulating factor-1 receptor (CSF-1R) Type II to lead to the clinical candidate JTE-952
Ikegashira, Kazutaka, Ikenogami, Taku, Yamasaki, Takayuki, Oka, Takahiro, Hase, Yasunori, Miyagawa, Naoki, Inagaki, Koji, Kawahara, Iichiro, Koga, Yoshihisa, Hashimoto, HiromasaLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2019.02.006
Date:
February, 2019
File:
PDF, 1.25 MB
english, 2019