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Discovery of Polypharmacological Melanocortin-3 and -4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a µM MC4R Partial Agonist
Fleming, Katlyn A., Freeman, Katie T., Powers, Mike D., Santos, Radleigh G., Debevec, Ginamarie, Giulianotti, Marc A., Houghten, Richard A., Doering, Skye R., Pinilla, Clemencia, Haskell-Luevano, CarrLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b00053
Date:
February, 2019
File:
PDF, 1.21 MB
english, 2019