Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid In Vivo Inactivation of Bruton's Tyrosine Kinase (BTK)
Watterson, Scott H., Liu, Qingjie, Beaudoin Bertrand, Myra, Batt, Douglas G., Li, Ling, Pattoli, Mark A., Skala, Stacey, Chen, Lihong, Obermeier, Mary T., Moore, Robin, Yang, Zheng, Vickery, Rodney, ELanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b00167
Date:
March, 2019
File:
PDF, 872 KB
english, 2019