Discovery and Lead-optimization of 4,5-Dihydropyrazoles as Mono-Kinase Selective, Orally Bioavailable and Efficacious Inhibitors of Receptor Interacting Protein 1 (RIP1) Kinase
Harris, Philip A., Faucher, Nicolas, George, Nicolas, Eidam, Patrick M, King, Bryan W., White, Gemma, Anderson, Niall A, Bandyopadhyay, Deepak, Beal, Allison M., BENETON, Veronique, Berger, Scott B.,Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b00318
Date:
April, 2019
File:
PDF, 1.82 MB
english, 2019