Identification of Diketopiperazine-Containing 2-Anilinobenzamides as Potent Sirtuin 2 (SIRT2)-Selective Inhibitors Targeting the “Selectivity Pocket”, Substrate-Binding Site, and NAD + -Binding Site
Mellini, Paolo, Itoh, Yukihiro, Elboray, Elghareeb E., Tsumoto, Hiroki, Li, Ying, Suzuki, Miki, Takahashi, Yukari, Tojo, Toshifumi, Kurohara, Takashi, Miyake, Yuka, Miura, Yuri, Kitao, Yuki, Kotoku, MLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b00255
Date:
May, 2019
File:
PDF, 1.59 MB
english, 2019