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Novel phenanthridin-6(5H)-one derivatives as potent and selective BET bromodomain inhibitors: Rational design, synthesis and biological evaluation
Zhi, Yanle, Wang, Shu, Huang, Wenhai, Zeng, Shenxin, Liang, Meihao, Zhang, Chixiao, Ma, Zhen, Wang, Zunyuan, Zhang, Zhimin, Shen, ZhengrongLanguage:
english
Journal:
European Journal of Medicinal Chemistry
DOI:
10.1016/j.ejmech.2019.06.067
Date:
June, 2019
File:
PDF, 1.26 MB
english, 2019