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Discovery of a First-in-Class Receptor Interacting Protein 2 (RIP2) Kinase Specific Clinical Candidate, 2-((4-(Benzo[ d ]thiazol-5-ylamino)-6-( tert -butylsulfonyl)quinazolin-7-yl)oxy)ethyl Dihydrogen Phosphate, for the Treatment of Inflammatory Diseases
Haile, Pamela A., Casillas, Linda N., Votta, Bartholomew J., Wang, Gren Z., Charnley, Adam K., Dong, Xiaoyang, Bury, Michael J., Romano, Joseph J., Mehlmann, John F., King, Bryan W., Erhard, Karl F.,Language:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b00575
Date:
July, 2019
File:
PDF, 2.95 MB
english, 2019