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SAR inspired by aldehyde oxidase (AO) metabolism: Discovery of novel, CNS penetrant tricyclic M4 PAMs
Chopko, Trevor C., Han, Changho, Gregro, Alison R., Engers, Darren W., Felts, Andrew S., Poslusney, Mike S., Bollinger, Katrina A., Morrison, Ryan D., Bubser, Michael, Lamsal, Atin, Luscombe, VincentJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2019.06.032
Date:
June, 2019
File:
PDF, 593 KB
2019