Structure-based and property-driven optimization of N-aryl imidazoles towards potent and selective oral RORγt inhibitors
Hoegenauer, Klemens, Kallen, Joerg, Jimenez-Nunez, Eloisa, Strang, Ross, Ertl, Peter, Cooke, Nigel G., Hintermann, Samuel, Voegtle, Markus, Betschart, Claudia, Mckay, Daniel J. J., Wagner, Juergen, OtLanguage:
english
Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b01291
Date:
November, 2019
File:
PDF, 967 KB
english, 2019