Discovery of structurally distinct tricyclic M4 positive allosteric modulator (PAM) chemotypes
Temple, Kayla J., Long, Madeline F., Engers, Julie L., Watson, Katherine J., Chang, Sichen, Luscombe, Vincent B., Rodriguez, Alice L., Niswender, Colleen M., Bridges, Thomas M., Jeffrey Conn, P., EngeLanguage:
english
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2019.126811
Date:
November, 2019
File:
PDF, 701 KB
english, 2019