Discovery of a novel 2,3-dimethylimidazo[1,2-a]pyrazine-6-carboxamide M4 positive allosteric modulator (PAM) chemotype
Temple, Kayla J., Engers, Julie L., Long, Madeline F., Watson, Katherine J., Chang, Sichen, Luscombe, Vincent B., Jenkins, Matthew T., Rodriguez, Alice L., Niswender, Colleen M., Bridges, Thomas M., JJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2019.126812
Date:
November, 2019
File:
PDF, 410 KB
2019