Discovery of Potent and Selective Antibody–Drug Conjugates with Eg5 Inhibitors through Linker and Payload Optimization
Karpov, Alexei S., Nieto-Oberhuber, Cristina M., Abrams, Tinya, Beng-Louka, Edwige, Blanco, Enrique, Chamoin, Sylvie, Chene, Patrick, Dacquignies, Isabelle, Daniel, Dylan, Dillon, Michael P., DoumampoJournal:
ACS Medicinal Chemistry Letters
DOI:
10.1021/acsmedchemlett.9b00468
Date:
December, 2019
File:
PDF, 1.50 MB
2019