Structure-activity relationship in pyrazolo[4,3-c]pyridines, first inhibitors of PEX14-PEX5 Protein-Protein Interaction (PPI) with trypanocidal activity
Dawidowski, Maciej, Kalel, Vishal C., Napolitano, Valeria, Fino, Roberto, Schorpp, Kenji, Emmanouilidis, Leonidas, Lenhart, Dominik, Ostertag, Michael, Kaiser, Marcel, Kolonko, Marta, Tippler, BettinaJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b01876
Date:
December, 2019
File:
PDF, 4.35 MB
2019