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Structure-based design of a potent and selective covalent inhibitor for SRC kinase that targets a p-Loop cysteine
Du, Guangyan, Rao, Suman, Gurbani, Deepak, Henning, Nathaniel J., Jiang, Jie, Che, Jianwei, Yang, Annan, Ficarro, Scott B, Marto, Jarrod A., Aguirre, Andrew J., Sorger, Peter K., Westover, Kenneth DalJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b01502
Date:
January, 2020
File:
PDF, 18.42 MB
2020