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Discovery of highly potent benzimidazole derivatives as indoleamine 2,3-dioxygenase-1 (IDO1) inhibitors: from structure-based virtual screening to in vivo pharmacodynamic activity
Serafini, Marta, Torre, Enza, Aprile, Silvio, Del Grosso, Erika, Gesù, Alessandro, Griglio, Alessia, Colombo, Giorgia, Travelli, Cristina, Paiella, Salvatore, Adamo, Annalisa, Orecchini, Elena, ColetJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.9b01809
Date:
March, 2020
File:
PDF, 1.11 MB
2020