Discovery of Orally Bioavailable Chromone Derivatives as Potent and Selective BRD4 Inhibitors: Scaffold Hopping, Optimization, and Pharmacological Evaluation
Liu, Zhiqing, Chen, Haiying, Wang, Pingyuan, Li, Yi, Wold, Eric A., Leonard, Paul G., Joseph, Sarah, Brasier, Allan R., Tian, Bing, Zhou, JiaJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00035
Date:
April, 2020
File:
PDF, 1.30 MB
2020