Fragment-based discovery of pyrazolopyridones as JAK1 inhibitors with excellent subtype selectivity
Hansen, Bettina Borreschmidt, Jepsen, Tue Heesgaard, Larsen, Mogens, Sindet, Rikke, Vifian, Thomas, Burhardt, Mia Nørreskov, Larsen, Jens, Seitzberg, Jimmi Gerner, Carnerup, Martin A, Jerre, Anders,Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00359
Date:
May, 2020
File:
PDF, 2.20 MB
2020