Bioisosteric Replacement of Arylamide-linked Spine Residues by N-Acylhydrazones and Selenophenes as Design Strategy to Novel Dibenzosuberone Derivatives as Type I½ p38ï¡ MAP Kinase Inhibitors
Galvez Bulhõ, es Pedreira, Jú, lia, Nahidino, Philipp, Kudolo, Mark, Pantsar, Tatu, Berger, Benedict-Tilman, Forster, Michael, Knapp, Stefan, Laufer, Stefan A., Barreiro, Eliezer J.Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00508
Date:
May, 2020
File:
PDF, 614 KB
2020