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Structure-Permeability Relationship of Semi-Peptidic Macrocycles â Understanding and Optimizing Passive Permeability and Efflux Ratio
Le Roux, Antoine, Blaise, Emilie, Boudreault, Pierre-Luc, Comeau, Christian, Doucet, Annie, Giarrusso, Marilena, Collin, Marie-Pierre, Neubauer, Thomas, Koelling, Florian, Göller, Andreas H., Seep, LJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00013
Date:
May, 2020
File:
PDF, 557 KB
2020