Design, synthesis and biological activity evaluation of novel 4-((1-cyclopropyl-3-(tetrahydro-2H-pyran-4-yl)-1H-pyrazol-4-yl) oxy) pyridine-2-yl) amino derivatives as potent transforming growth factor-β (TGF-β) type I receptor inhibitors
Tan, Bin, Zhang, Xiaomeng, Quan, Xu, Zheng, Guochuang, Li, Xue, Zhao, Liwen, Li, Wei, Li, BoJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2020.127339
Date:
June, 2020
File:
PDF, 715 KB
2020