Design, synthesis and biological evaluation of novel 6-phenyl-1,3a,4,10b-tetrahydro-2H-benzo[c]thiazolo[4,5-e]azepin-2-one derivatives as potential BRD4 inhibitors
Li, Qifei, Li, Jieming, Cai, Yan, Zou, Yuxing, Chen, Bin, Zou, Feng, Mo, Jiaxian, Han, Ting, Guo, Weiwei, Huang, Wenlong, Qiu, Qianqian, Qian, HaiVolume:
28
Journal:
Bioorganic & Medicinal Chemistry
DOI:
10.1016/j.bmc.2020.115601
Date:
August, 2020
File:
PDF, 4.16 MB
2020