Discovery of (3S,4S)-3-methyl-3-(4-fluorophenyl)-4-(4-(1,1,1,3,3,3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines as novel RORγt inverse agonists
Jiang, Bin, Duan, James J.W., Stachura, Sylwia, Karmakar, Ananta, Hemagiri, Hemalatha, Kumar Raut, Dhanya, Kumar Gupta, Arun, Weigelt, Carolyn A., Khan, Javed, Sack, John S., Wu, Dauh-Rurng, Yarde, MeJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2020.127392
Date:
July, 2020
File:
PDF, 836 KB
2020