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The Optimisation of a Novel, Weak Bromo and Extra Terminal Domain (BET) Bromodomain Fragment Ligand to a Potent and Selective Second Bromodomain (BD2) Inhibitor
Seal, Jonathan Thomas, Atkinson, Stephen J., Aylott, Helen, Bamborough, Paul, Chung, Chun-wa, Copley, Royston C. B., Gordon, Laurie J., Grandi, Paola, Gray, James R. J., Harrison, Lee A, Hayhow, ThomaJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00796
Date:
July, 2020
File:
PDF, 1.05 MB
2020