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Structure-Based Design of a Bromodomain and Extraterminal Domain (BET) Inhibitor Selective for the N-Terminal Bromodomains That Retains an Anti-inflammatory and Antiproliferative Phenotype
Wellaway, Christopher R., Bamborough, Paul, Bernard, Sharon G., Chung, Chun-wa, Craggs, Peter D., Cutler, Leanne, Demont, Emmanuel H., Evans, John P., Gordon, Laurie, Karamshi, Bhumika, Lewis, AntoniaJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00566
Date:
August, 2020
File:
PDF, 6.80 MB
2020