Discovery of substituted 3H-pyrido[2,3-d]pyrimidin-4-ones as potent, biased, and orally bioavailable sst2 agonist
Zhao, Jian, Chen, Zhiyong, Kusnetzow, Ana Karin, Nguyen, Julie, Rico-Bautista, Elizabeth, Tan, Hannah, Betz, Stephen F., Struthers, R. Scott, Zhu, YunfeiJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2020.127496
Date:
August, 2020
File:
PDF, 448 KB
2020