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Discovery of PROTAC molecules that selectively degrade the IRAK3 pseudokinase.
Degorce, Sebastien L., Tavana, Omid, Banks, Erica, Crafter, Claire, Gingipalli, Lakshmaiah, Kouvchinov, David, Mao, Yumeng, Pachl, Fiona, Solanki, Anisha, Valge-Archer, Viia, Yang, Bin, Edmondson, ScoJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c01125
Date:
August, 2020
File:
PDF, 4.53 MB
2020