Highly selective sub-nanomolar cathepsin S inhibitors by merging fragment binders with covalent nitrile inhibitors
Schade, Markus, Merla, Beatrix, Lesch, Bernhard, Wagener, Markus, Timmermanns, Simone, Pletinckx, Katrien, Hertrampf, TorstenJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c00949
Date:
September, 2020
File:
PDF, 635 KB
2020