Discovery of AZD9833, a potent and orally bioavailable selective estrogen receptor degrader and antagonist.
Scott, James S., Moss, Thomas A., Balazs, Amber, Barlaam, Bernard, Breed, Jason, Carbajo, Rodrigo, Chiarparin, Elisabetta, Davey, Paul, Delpuech, Oona, Fawell, Stephen, Fisher, David, gagrica, sladjanJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c01163
Date:
September, 2020
File:
PDF, 1.27 MB
2020