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Torin 2 derivative, NCATS-SM3710, has potent multistage antimalarial activity through inhibition of P. falciparum phosphatidylinositol 4-kinase (Pf PI4KIIIβ)
Krishnan, Karthik, Ziniel, Peter, Li, Hao, Huang, Xiuli, Hupalo, Daniel, Gombakomba, Nita, Mendoza Guerrero, Sandra, Dotrang, Thoai, Lu, Xiao, Caridha, Diana, Sternberg, Anna R., Hughes, Emma, Sun, WeJournal:
ACS Pharmacology & Translational Science
DOI:
10.1021/acsptsci.0c00078
Date:
September, 2020
File:
PDF, 885 KB
2020