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A two-tiered in vitro approach to de-risk drug candidates for potential bile salt export pump inhibition liabilities in drug discovery
Hafey, Michael J., Houle, Robert, Tanis, Keith Q., Knemeyer, Ian, Shang, Jackie, Chen, Qing, Baudy, Andreas, Monroe, James, Sistare, Frank D., Evers, RaymondJournal:
Drug Metabolism and Disposition
DOI:
10.1124/dmd.120.000086
Date:
September, 2020
File:
PDF, 1.83 MB
2020