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Structure-based optimisation of orally active & reversible MetAP-2 inhibitors maintaining a tight âmolecular budgetâ
Hirst, David J., Brandt, Martin, Bruton, Gordon, Christodoulou, Erica, Cutler, Leanne, Deeks, Nigel, Goodacre, Jonathan D., Jack, Torquil, Lindon, Matthew, Miah, Afjal, Page, Kevin, Parr, Nigel, ShuklJournal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2020.127533
Date:
September, 2020
File:
PDF, 1.77 MB
2020