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Discovery of 1-(1H-indazol-4-yl)-3-((1-phenyl-1H-pyrazol-5-yl)methyl) ureas as potent and thermoneutral TRPV1 antagonists
Kang, Jin Mi, Kwon, Sun Ok, Ann, Jihyae, Blumberg, Peter M., Ha, Heejin, Yoo, Young Dong, Frank-Foltyn, Robert, Lesch, Bernhard, Bahrenberg, Gregor, Stockhausen, Hannelore, Christoph, Thomas, Lee, JeeVolume:
30
Journal:
Bioorganic & Medicinal Chemistry Letters
DOI:
10.1016/j.bmcl.2020.127548
Date:
December, 2020
File:
PDF, 667 KB
2020