Predicting the Permeability of Macrocycles from Conformational Sampling â Limitations of Molecular Flexibility
Poongavanam, Vasanthanathan, Atilaw, Yoseph, Ye, Sofie, Wieske, Lianne H.E., Erdelyi, Mate, Ermondi, Giuseppe, Caron, Giulia, Kihlberg, JanJournal:
Journal of Pharmaceutical Sciences
DOI:
10.1016/j.xphs.2020.10.052
Date:
October, 2020
File:
PDF, 6.33 MB
2020