From Pyrazolones to Azaindoles: Evolution of Active-Site SHP2 Inhibitors Based on Scaffold Hopping and Bioisosteric Replacement
Mostinski, Yelena, Heynen, Guus J. J. E., López-Alberca, Maria Pascual, Paul, Jerome, Miksche, Sandra, Radetzki, Silke, Schaller, David, Shanina, Elena, Seyffarth, Carola, Kolomeets, Yuliya, Ziebart,Journal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c01265
Date:
November, 2020
File:
PDF, 4.81 MB
2020