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A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation
Picado, Alfredo, Chaikuad, Apirat, Wells, Carrow I., Shrestha, Safal, Zuercher, William J., Pickett, Julie E., Kwarcinski, Frank E., Sinha, Parvathi, de Silva, Chandi S., Zutshi, Reena, Liu, Shubin, KJournal:
Journal of Medicinal Chemistry
DOI:
10.1021/acs.jmedchem.0c01174
Date:
November, 2020
File:
PDF, 6.96 MB
2020