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Volume 31; Issue 3
Main
Investigational New Drugs
Volume 31; Issue 3
Investigational New Drugs
Volume 31; Issue 3
1
Phase 2 study of carlumab (CNTO 888), a human monoclonal antibody against CC-chemokine ligand 2 (CCL2), in metastatic castration-resistant prostate cancer
Pienta, Kenneth J.
,
Machiels, Jean-Pascal
,
Schrijvers, Dirk
,
Alekseev, Boris
,
Shkolnik, Mikhail
,
Crabb, Simon J.
,
Li, Susan
,
Seetharam, Shobha
,
Puchalski, Thomas A.
,
Takimoto, Chris
,
Elsayed, Yusri
,
D
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 232 KB
Your tags:
english, 2013
2
Expression of matrix macromolecules and functional properties of EGF-responsive colon cancer cells are inhibited by panitumumab
Gialeli, Ch.
,
Theocharis, A. D.
,
Kletsas, D.
,
Tzanakakis, G. N.
,
Karamanos, N. K.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 551 KB
Your tags:
english, 2013
3
A novel proteasome inhibitor acting in mitochondrial dysfunction, ER stress and ROS production
Maria, Durvanei Augusto
,
Souza, Jean Gabriel
,
Morais, Katia L. P.
,
Berra, Carolina Maria
,
Zampolli, Hamilton de Campos
,
Demasi, Marilene
,
Simons, Simone Michaela
,
Freitas Saito, Renata
,
Chammas, Roger
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 631 KB
Your tags:
english, 2013
4
Gambogic acid is cytotoxic to cancer cells through inhibition of the ubiquitin-proteasome system
Felth, Jenny
,
Lesiak-Mieczkowska, Karolina
,
DâArcy, Padraig
,
Haglund, Caroline
,
Gullbo, Joachim
,
Larsson, Rolf
,
Linder, Stig
,
Bohlin, Lars
,
Fryknäs, Mårten
,
Rickardson, Linda
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 532 KB
Your tags:
english, 2013
5
Cytotoxicity of withaferin A in glioblastomas involves induction of an oxidative stress-mediated heat shock response while altering Akt/mTOR and MAPK signaling pathways
Grogan, Patrick T.
,
Sleder, Kristina D.
,
Samadi, Abbas K.
,
Zhang, Huaping
,
Timmermann, Barbara N.
,
Cohen, Mark S.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 981 KB
Your tags:
english, 2013
6
A phase I study of IMP321 and gemcitabine as the front-line therapy in patients with advanced pancreatic adenocarcinoma
Wang-Gillam, Andrea
,
Plambeck-Suess, Stacey
,
Goedegebuure, Peter
,
Simon, Peter O.
,
Mitchem, Jonathan B.
,
Hornick, John R.
,
Sorscher, Steven
,
Picus, Joel
,
Suresh, Rama
,
Lockhart, Albert C.
,
Tan, Benjam
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 174 KB
Your tags:
english, 2013
7
EGFR and HER2 inhibition in pancreatic cancer
Walsh, Naomi
,
Kennedy, Susan
,
Larkin, AnneMarie
,
Corkery, Brendan
,
O’Driscoll, Lorraine
,
Clynes, Martin
,
Crown, John
,
O’Donovan, Norma
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 576 KB
Your tags:
english, 2013
8
Dual modulation of JNK and Akt signaling pathways by chaetoglobosin K in human lung carcinoma andras-transformed epithelial cells
Ali, Amna
,
Sidorova, Tatyana S.
,
Matesic, Diane F.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 583 KB
Your tags:
english, 2013
9
The novel antiangiogenic VJ115 inhibits the NADH oxidase ENOX1 and cytoskeleton-remodeling proteins
Venkateswaran, Amudhan
,
Friedman, David B.
,
Walsh, Alexandra J.
,
Skala, Melissa C.
,
Sasi, Soumya
,
Rachakonda, Girish
,
Crooks, Peter A.
,
Freeman, Michael L.
,
Sekhar, Konjeti R.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 582 KB
Your tags:
english, 2013
10
A Phase 1 dose-escalation study of the safety and pharmacokinetics of once-daily oral foretinib, a multi-kinase inhibitor, in patients with solid tumors
Shapiro, Geoffrey I.
,
McCallum, Stewart
,
Adams, Laurel M.
,
Sherman, Laurie
,
Weller, Steve
,
Swann, Suzanne
,
Keer, Harold
,
Miles, Dale
,
Müller, Thomas
,
LoRusso, Patricia
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 260 KB
Your tags:
english, 2013
11
Phase I and pharmacokinetic study of pazopanib and lapatinib combination therapy in patients with advanced solid tumors
Jonge, Maja J. A.
,
Hamberg, Paul
,
Verweij, Jaap
,
Savage, Shawna
,
Suttle, A. Benjamin
,
Hodge, Jeffrey
,
Arumugham, Thangam
,
Pandite, Lini N.
,
Hurwitz, Herbert I.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 165 KB
Your tags:
english, 2013
12
A phase 1 study of TRC102, an inhibitor of base excision repair, and pemetrexed in patients with advanced solid tumors
Gordon, Michael S.
,
Rosen, Lee S.
,
Mendelson, David
,
Ramanathan, Ramesh K.
,
Goldman, Jonathan
,
Liu, Lili
,
Xu, Yan
,
Gerson, Stanton L.
,
Anthony, Stephen P.
,
Figg, William D.
,
Spencer, Shawn
,
Adams, Bon
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 224 KB
Your tags:
english, 2013
13
Phase I and pharmacokinetic study of IV vinflunine in cancer patients with liver dysfunction
Delord, J. P.
,
Ravaud, A.
,
Bennouna, J.
,
Fumoleau, P.
,
Favrel, S.
,
Pinel, M. C.
,
Ferré, P.
,
Saliba, F.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 255 KB
Your tags:
english, 2013
14
A pilot study for the early assessment of the effects of BMS-754807 plus gefitinib in an H292 tumor model by [18F]fluorothymidine-positron emission tomography
Lee, Seung Jin
,
Kim, Eun Jung
,
Lee, Haeng Jung
,
Kim, Seog Young
,
Oh, Seung Jun
,
Ryu, Jin Sook
,
Moon, Dae Hyuk
,
Ahn, Jin-Hee
,
Kim, Sang-We
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 531 KB
Your tags:
english, 2013
15
The risk of hand-foot skin reaction to axitinib, a novel VEGF inhibitor: a systematic review of literature and meta-analysis
Fischer, Alyssa
,
Wu, Shenhong
,
Ho, Alan L.
,
Lacouture, Mario E.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 284 KB
Your tags:
english, 2013
16
Characterization of a membrane-active anti-tumor agent, UA8967
Dorr, Robert T.
,
Samulitis, Betty K.
,
Wisner, Lee
,
Han, Haiyong
,
Zhao, Yu
,
Beroza, Paul
,
Damodaran, Komath
,
Igarashi, Suzu
,
Landowski, Terry H.
,
Hoff, Daniel D.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 673 KB
Your tags:
english, 2013
17
Erratum to: Safety and tolerability of AZD8055 in Japanese patients with advanced solid tumors; a dose-finding phase I study
Asahina, Hajime
,
Nokihara, Hiroshi
,
Yamamoto, Noboru
,
Yamada, Yasuhide
,
Tamura, Yosuke
,
Honda, Kazunori
,
Seki, Yoshitaka
,
Tanabe, Yuko
,
Shimada, Hitoshi
,
Shi, Xiaojin
,
Tamura, Tomohide
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 187 KB
Your tags:
english, 2013
18
Phase I study of pulsatile 3-day administration of afatinib (BIBW 2992) in combination with docetaxel in advanced solid tumors
Awada, A. H.
,
Dumez, H.
,
Hendlisz, A.
,
Wolter, P.
,
Besse-Hammer, T.
,
Uttenreuther-Fischer, M.
,
Stopfer, P.
,
Fleischer, F.
,
Piccart, M.
,
Schöffski, P.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 269 KB
Your tags:
english, 2013
19
Sorafenibinhibits in vitro osteoclastogenesis by down-modulating Mcl-1
Rimondi, Erika
,
Secchiero, Paola
,
Melloni, Elisabetta
,
Grill, Vittorio
,
Zauli, Giorgio
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 396 KB
Your tags:
english, 2013
20
Phase II study of the Src kinase inhibitor saracatinib (AZD0530) in metastatic melanoma
Gangadhar, Tara C.
,
Clark, Joseph I.
,
Karrison, Theodore
,
Gajewski, Thomas F.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 146 KB
Your tags:
english, 2013
21
Preclinical evaluation of the AKT inhibitor MK-2206 in nasopharyngeal carcinoma cell lines
Ma, Brigette B. Y.
,
Lui, Vivian W. Y.
,
Hui, Connie W. C.
,
Lau, Cecilia P. Y.
,
Wong, Chi-Hang
,
Hui, Edwin P.
,
Ng, Margaret H.
,
Tsao, S. W.
,
Li, Yan
,
Chan, Anthony T. C.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 691 KB
Your tags:
english, 2013
22
Determinants of patient screen failures in Phase 1 clinical trials
Mckane, Alexandra
,
Sima, Chao
,
Ramanathan, Ramesh K.
,
Jameson, Gayle
,
Mast, Cathy
,
White, Erica
,
Fleck, Sharon
,
Downhour, Molly
,
Hoff, Daniel D.
,
Weiss, Glen J.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 217 KB
Your tags:
english, 2013
23
Metabolism of patupilone in patients with advanced solid tumor malignancies
Kelly, Kevin R.
,
Zollinger, Markus
,
Lozac’h, Frédéric
,
Tan, Eugene
,
Mita, Alain
,
Waldmeier, Felix
,
Urban, Patrick
,
Anand, Suraj
,
Wang, Yanfeng
,
Swart, Piet
,
Takimoto, Chris
,
Mita, Monica
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 285 KB
Your tags:
english, 2013
24
Phase I study of enzastaurin and bevacizumab in patients with advanced cancer: safety, efficacy and pharmacokinetics
Nwankwo, Nwabundo
,
Zhang, Zhe
,
Wang, Ting
,
Collins, Connie
,
Resta, Lee
,
Ermisch, Sabine
,
Day, Jeannette
,
Decker, Rodney
,
Kornberg, Lori
,
Nicol, Steven
,
Thornton, Donald
,
Armstrong, Deborah K.
,
Carducc
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 344 KB
Your tags:
english, 2013
25
Phase I study of matuzumab in combination with 5-fluorouracil, leucovorin and cisplatin (PLF) in patients with advanced gastric and esophagogastric adenocarcinomas
Trarbach, Tanja
,
Przyborek, Marta
,
Schleucher, Norbert
,
Heeger, Steffen
,
Lüpfert, Christian
,
Vanhoefer, Udo
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 269 KB
Your tags:
english, 2013
26
A phase IB trial of 24-hour intravenous PX-12, a thioredoxin-1 inhibitor, in patients with advanced gastrointestinal cancers
Baker, A. F.
,
Adab, K. N.
,
Raghunand, N.
,
Chow, H. H. S.
,
Stratton, S. P.
,
Squire, S. W.
,
Boice, M.
,
Pestano, L. A.
,
Kirkpatrick, D. L.
,
Dragovich, T.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 426 KB
Your tags:
english, 2013
27
A phase I study of DHP107, a mucoadhesive lipid form of oral paclitaxel, in patients with advanced solid tumors: Crossover comparisons with intravenous paclitaxel
Hong, Yong Sang
,
Kim, Kyu-pyo
,
Lim, Hyeong-Seok
,
Bae, Kyun-Seop
,
Ryu, Min-Hee
,
Lee, Jae-Lyun
,
Chang, Heung Moon
,
Kang, Yoon-Koo
,
Kim, Hyeyoun
,
Kim, Tae Won
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 198 KB
Your tags:
english, 2013
28
Phase I study of PM00104 (Zalypsis®) administered as a 1-hour weekly infusion resting every fourth week in patients with advanced solid tumors
Massard, Christophe
,
Margetts, Jane
,
Amellal, Nadia
,
Drew, Yvette
,
Bahleda, Ratislav
,
Stevens, Peter
,
Armand, Jean Pierre
,
Calvert, Hilary
,
Soria, Jean Charles
,
Coronado, Cinthya
,
Kahatt, Carmen
,
Alfa
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 171 KB
Your tags:
english, 2013
29
A phase I study of S-1 with concurrent radiotherapy in elderly patients with locally advanced non-small cell lung cancer
Hasegawa, Yoshikazu
,
Okamoto, Isamu
,
Takezawa, Ken
,
Miyazaki, Masaaki
,
Tsurutani, Junji
,
Yonesaka, Kimio
,
Morinaga, Ryotaroh
,
Tsuya, Asuka
,
Terashima, Masaaki
,
Kudoh, Toshihiro
,
Azuma, Koichi
,
Kurata,
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 201 KB
Your tags:
english, 2013
30
REO-001: A phase I trial of percutaneous intralesional administration of reovirus type 3 dearing (Reolysin®) in patients with advanced solid tumors
Morris, Don G.
,
Feng, Xiaolan
,
DiFrancesco, Lisa M.
,
Fonseca, Kevin
,
Forsyth, Peter A
,
Paterson, Alexander H.
,
Coffey, Matt C.
,
Thompson, Brad
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 236 KB
Your tags:
english, 2013
31
A phase I study of prolonged infusion of triapine in combination with fixed dose rate gemcitabine in patients with advanced solid tumors
Mortazavi, Amir
,
Ling, Yonghua
,
Martin, Ludmila Katherine
,
Wei, Lai
,
Phelps, Mitch A.
,
Liu, Zhongfa
,
Harper, Erica J.
,
Ivy, S. Percy
,
Wu, Xin
,
Zhou, Bing-Sen
,
Liu, Xiyong
,
Deam, Deidre
,
Monk, J. Paul
,
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 240 KB
Your tags:
english, 2013
32
Safety and tolerability of AZD8055 in Japanese patients with advanced solid tumors; a dose-finding phase I study
Asahina, Hajime
,
Nokihara, Hiroshi
,
Yamamoto, Noboru
,
Yamada, Yasuhide
,
Tamura, Yosuke
,
Honda, Kazunori
,
Seki, Yoshitaka
,
Tanabe, Yuko
,
Shimada, Hitoshi
,
Shi, Xiaojin
,
Tamura, Tomohide
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 317 KB
Your tags:
english, 2013
33
A phase I pharmacokinetic study of matuzumab in combination with paclitaxel in patients with EGFR-expressing advanced non-small cell lung cancer
Hartmann, J. T.
,
Kollmannsberger, C.
,
Cascorbi, I.
,
Mayer, F.
,
Schittenhelm, M. M.
,
Heeger, S.
,
Bokemeyer, C.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 151 KB
Your tags:
english, 2013
34
A phase 1 study of a chimeric monoclonal antibody against interleukin-6, siltuximab, combined with docetaxel in patients with metastatic castration-resistant prostate cancer
Hudes, Gary
,
Tagawa, Scott T.
,
Whang, Young E.
,
Qi, Ming
,
Qin, Xiang
,
Puchalski, Thomas A.
,
Reddy, Manjula
,
Cornfeld, Mark
,
Eisenberger, Mario
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 208 KB
Your tags:
english, 2013
35
Erratum to: Phase I study of PM00104 (Zalypsis®) administered as a 1-hour weekly infusion resting every fourth week in patients with advanced solid tumors
Massard, Christophe
,
Margetts, Jane
,
Amellal, Nadia
,
Drew, Yvette
,
Bahleda, Ratislav
,
Stephens, Peter
,
Armand, Jean Pierre
,
Calvert, Hilary
,
Soria, Jean Charles
,
Coronado, Cinthya
,
Kahatt, Carmen
,
Alf
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 49 KB
Your tags:
english, 2013
36
Erratum to: Effect of the drug transporters ABCG2, Abcg2, ABCB1 and ABCC2 on the disposition, brain accumulation and myelotoxicity of the aurora kinase B inhibitor barasertib and its more active form barasertib-hydroxy-QPA
Marchetti, Serena
,
Pluim, Dick
,
Eijndhoven, Monique
,
Tellingen, Olaf
,
Mazzanti, Roberto
,
Beijnen, Jos H.
,
Schellens, Jan H. M.
Journal:
Investigational New Drugs
Year:
2013
Language:
english
File:
PDF, 47 KB
Your tags:
english, 2013
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