Volume 24; Issue 1

Journal of Medicinal Chemistry

Volume 24; Issue 1

1

Synthesis and angiotensin-converting enzyme inhibitory activity of 3-(mercaptomethyl)-2-oxo-1-pyrrolidineacetic acids and 3-(mercaptomethyl)-2-oxo-1-piperidineacetic acids

Klutchko, Sylvester, Hoefle, Milton L., Smith, Ronald D., Essenburg, Arnold D., Parker, Robert B., Nemeth, Vicki L., Ryan, Michael, Dugan, Deborah H., Kaplan, Harvey R.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 823 KB

english, 1981

2

Synthesis and antihypertensive activity of new 6-heteroaryl-3-hydrazinopyridazine derivatives

Steiner, Gerd, Gries, Josef, Lenke, Dieter

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 647 KB

english, 1981

3

Piperazinylquinoxalines with central serotoninmimetic activity

Lumma, William C., Hartman, Richard D., Saari, Walfred S., Engelhardt, Edward L., Lotti, Victor J., Stone, Clement A.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 1.04 MB

english, 1981

4

Importance of the aromatic ring in adrenergic amines. 5. Nonaromatic analogs of phenylethanolamine as inhibitors of phenylethanolamine N-methyltransferase: role of hydrophobic and steric interactions

Vincek, William C., Aldrich, Constance S., Borchardt, Ronald T., Grunewald, Gary L.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 836 KB

english, 1981

5

Synthesis and stereochemistry of 7-phenyl-2-propionanilidobenzo[a]quinolizidine derivatives. Structural probes of fentanyl analgesics

Maryanoff, Bruce E., McComsey, David F., Taylor, Russell J., Gardocki, Joseph F.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 1.43 MB

english, 1981

6

Toward more selective antiarthritic therapy

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 2.17 MB

english, 1981

7

Fluorinated retinoic acids and their analogs. 2. Synthesis and biological activity of aromatic 4-fluoro analogs

Chan, Ka-Kong, Specian, Anthony C., Pawson, Beverly A.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 556 KB

english, 1981

8

1-Oxacephalosporins: enhancement of .beta.-lactam reactivity and antibacterial activity

Murakami, Kazuhisa, Takasuka, Mamoru, Motokawa, Kiyoshi, Yoshida, Tadashi

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 769 KB

english, 1981

9

Tetrahydro-2-benzoxepins: a novel family of hypotensives

TenBrink, Ruth E., McCall, John M., Pals, Donald T., McCall, Robert B., Orley, John, Humphrey, Steve J., Wendling, Michael G.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 490 KB

english, 1981

10

Regiospecific attack of nitrogen and sulfur nucleophiles on quinones derived from poison oak/ivy catechols (urushiols) and analogs as models for urushiol-protein conjugate formation

Liberato, Daniel J., Byers, Vera S., Dennick, Reg G., Castagnoli, Neal

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 819 KB

english, 1981

11

New antiarrhythmic agents. 5. .alpha.-Aminoaceto-2,6-xylidides with functionalized amide alkyl substituents

McMaster, Paul D., Byrnes, Eugene W., Block, Alan J., Tenthorey, Paul A.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 913 KB

english, 1981

12

Masthead

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 240 KB

english, 1981

13

.alpha.-Ethynyl and .alpha.-vinyl analogs of ornithine as enzyme-activated inhibitors of mammalian ornithine decarboxylase

Danzin, Charles, Casara, Patrick, Claverie, Nicole, Metcalf, Brian W.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 716 KB

english, 1981

14

New antiarrhythmic agents. 4. 1'-(aminoalkyl)-1,2,3,4-tetrahydronaphthalene-1-spiro-3'-pyrrolidine-2',5'-dione derivatives

Tenthorey, Paul A., Ronfeld, Robert A., Feldman, Hal S., Sandberg, Rune V., McMaster, Paul D., Smith, Emil R.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 799 KB

english, 1981

15

Nonsteroidal antiinflammatroy agents. 2. Synthesis of 4',5-disubstituted 3-diphenylylacetic acids and their derivatives with antiinflammatory and analgesic activities

Tamura, Yasumitsu, Yoshimoto, Yoshihiko, Kunimoto, Katsutoshi, Tada, Shinichi, Matsumura, Shingo, Murayama, Masao, Shibata, Yoshihisa, Enomoto, Hiroshi

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 645 KB

english, 1981

16

2-(Aminomethyl)phenols, a new class of saluretic agents. 2. Synthesis and pharmacological properties of the 5-aza isostere of 2-(aminomethyl)-4-(1,1-dimethylethyl)-6-iodophenol

Stokker, G. E., Smith, R. L., Cragoe, E. J., Ludden, C. T., Russo, H. F., Sweet, C. S., Watson, L. S.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 361 KB

english, 1981

17

Synthesis and antiinflammatory activity of metabolites of piroxicam

Lombardino, Joseph G.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 480 KB

english, 1981

18

Synthesis and study of the potential antiallergic activity of some pyrazole derivatives

Di Parsia, Maria T., Suarez, Cecilia, Vitolo, Maria J., Marquez, Victor E., Beyer, Bernardo, Urbina, Cecilia, Hurtado, Ines

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 364 KB

english, 1981

19

Novel tetracyclic spiropiperidines. 1. 3-Aryl-1,3-dihydrospiro[benzo[c]thiophene-1,4'-piperidines] as potential antidepressants

Ong, Helen H., Profitt, James A., Anderson, V. Brian, Kruse, Hansjoerg, Wilker, Jeffrey C., Geyer, Harry M.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 699 KB

english, 1981

20

Book Reviews

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 138 KB

english, 1981

21

1-(Naphthylalkyl)-1H-imidazole derivatives, a new class of anticonvulsant agents

Walker, Keith A. M., Wallach, Marshall B., Hirschfeld, Donald R.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 870 KB

english, 1981

22

Synthesis of 2'-deoxy-L-fucopyranosylcarminomycinone and -.epsilon.-pyrromycinone as well as 2'-deoxy-D-erythro-pentopyranosyldaunomycinone, -carminomycinone, and -.epsilon.-pyrromycinone

El Khadem, Hassan S., Swartz, David L.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 450 KB

english, 1981

23

Importance of the aromatic ring in adrenergic amines. 6. Nonaromatic analogs of phenylethanolamine as inhibitors of phenylethanolamine N-methyltransferase: role of .pi.-electronic and steric interactions

Davis, Dwight P., Borchardt, Ronald T., Grunewald, Gary L.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 727 KB

english, 1981

24

Synthesis and antiviral activity of 1-(2-deoxy-.beta.-D-ribofuranosyl)-5-(methylmercapto)-2-pyrimidinone

Schroeder, Alan C., Bardos, Thomas J., Cheng, Yung-Chi

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 569 KB

english, 1981

25

Permethyl analog of the pyrrolic antibiotic distamycin A

Gendler, Paul L., Rapoport, Henry

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 888 KB

english, 1981

26

Novel peptidoaminobenzophenones, terminal N-substituted peptidoaminobenzophenones, and N-(acylglycyl)aminobenzophenones as open-ring derivatives of benzodiazepines

Hirai, Kentaro, Ishiba, Teruyuki, Sugimoto, Hirohiko, Fujishita, Toshio, Tsukinoki, Yuji, Hirose, Katsumi

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 917 KB

english, 1981

27

Potential organ- or tumor-imaging agents. 21. Acyl-labeled esters of cholesterol

Counsell, R. E., Seevers, R. H., Korn, N., Schwendner, S. W.

Journal:

Journal of Medicinal Chemistry

Year:

1981

Language:

english

File:

PDF, 230 KB

english, 1981

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