Volume 28; Issue 11

Journal of Medicinal Chemistry

Volume 28; Issue 11

1

Potential antitumor agents. 44. Synthesis and antitumor activity of new classes of diacridines: importance of linker chain rigidity for DNA binding kinetics and biological activity

Denny, William A., Atwell, Graham J., Baguley, Bruce C., Wakelin, Laurence P. G.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 994 KB

english, 1985

2

Antitrichomonal activity of mesoionic thiazolo[3,2-a]pyridines

Walker, Keith A. M., Sjogren, Eric B., Matthews, Thomas R.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 813 KB

english, 1985

3

Opioid receptor interactions and conformations of the 6.alpha. and 6.beta. epimers of oxymorphamine. Solid-state conformation of 6.alpha.-oxymorphamine

Lever, O. William, Bhatia, Ashok V., Chang, Kwen Jen

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 671 KB

english, 1985

4

Imidazo[1,5-d][1,2,4]triazines as potential antiasthma agents

Paul, Rolf, Brockman, John A., Hallett, W. A., Hanifin, John W., Tarrant, M. Ernestine, Torley, Lawrence W., Callahan, Francis M., Fabio, Paul F., Johnson, Bernard D.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.49 MB

english, 1985

5

Synthesis of 6-anilino-2-thiouracils and their inhibition of human placenta iodothyronine deiodinase

Emerson, C. H., Braverman, L. E., Wu, C. F., Gambino, J., Wright, G. E., Nogimori, T.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 472 KB

english, 1985

6

5-(Haloalkyl)-2'-deoxyuridines: a novel type of potent antiviral nucleoside analog

Griengl, Herfried, Bodenteich, Michael, Hayden, Walter, Wanek, Erich, Streicher, Wolfgang, Stuetz, Peter, Bachmayer, Helmut, Ghazzouli, Ismail, Rosenwirth, Brigitte

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 812 KB

english, 1985

7

Pseudosymmetry and bioisosterism in biaryl pyridyl competitive histamine H2-receptor antagonists

Lipinski, Christopher A., LaMattina, John L., Hohnke, Lyle A.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.15 MB

english, 1985

8

N-(Phosphonoacetyl)amino phosphonates. Phosphonate analogs of N-(phosphonoacetyl)-L-aspartic acid (PALA)

Kafarski, Pawel, Lejczak, Barbara, Mastalerz, Przemyslaw, Dus, Danuta, Radzikowski, Czeslaw

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 500 KB

english, 1985

9

Hypolipidemic activity of indan-1,3-dione derivatives in rodents

Murthy, A. R., Wyrick, S. D., Hall, I. H.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 785 KB

english, 1985

10

Design and synthesis of new transition-state analog inhibitors of aspartate transcarbamylase

Farrington, G. King, Kumar, Alok, Wedler, Frederick C.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 908 KB

english, 1985

11

4-Substituted 5-[m-(trifluoromethyl)phenoxy]primaquine analogs as potential antimalarial agents

Carroll, F. Ivy, Berrang, Bertold, Linn, C. P.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 570 KB

english, 1985

12

Synthesis and structure-activity relationships of novel arylfluoroquinolone antibacterial agents

Chu, Daniel T. W., Fernandes, Prabhavathi B., Claiborne, Akiyo K., Pihuleac, Eva, Nordeen, Carl W., Maleczka, Robert E., Pernet, Andre G.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 872 KB

english, 1985

13

Novel nonnarcotic analgesics with an improved therapeutic ratio. Structure-activity relationships of 8-(methylthio)- and 8-(acylthio)-1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines

Hori, Mikio, Ban, Masatoshi, Imai, Eiji, Iwata, Noriyuki, Suzuki, Yoshinari, Baba, Yutaka, Morita, Tokiko, Fujimura, Hajime, Nozaki, Masakatsu, Niwa, Masayuki

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 756 KB

english, 1985

14

Synthesis and anthelmintic activity of 5(6)-[(benzimidazol-2-yl)carboxamido]- and (4-substituted piperazin-1-yl)benzimidazoles

Dubey, Rashmi, Abuzar, Syed, Sharma, Satyavan, Chatterjee, R. K., Katiyar, J. C.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 435 KB

english, 1985

15

Synthesis and antidiarrheal activity of N-(aminoiminomethyl)-1H-pyrrole-1-acetamides related to guanfacine

Beattie, Doreen E., Dover, Gillian M., Ward, Terence J.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 481 KB

english, 1985

16

.beta.-Adrenoceptor activity of the stereoisomers of the bufuralol alcohol and ketone metabolites

Machin, Peter J., Hurst, David N., Osbond, John M.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 525 KB

english, 1985

17

Synthesis and properties of bis(2,2-dimethylaziridinyl)phosphinic amides: a series of new antineoplastic agents

MacDiarmid, Joan E., Rose, William C., Biddle, William C., Perlman, Michael E., Breiner, Robert G., Ambrus, Julian L., Bardos, Thomas J.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 969 KB

english, 1985

18

Synthesis, absolute configuration and conformation of the aldose reductase inhibitor sorbinil

Sarges, Reinhard, Bordner, Jon, Dominy, Beryl W., Peterson, Michael J., Whipple, Earl B.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 558 KB

english, 1985

19

Angiotensin converting enzyme inhibitors: structure-activity profile of 1-benzazepin-2-one derivatives

Stanton, James L., Watthey, Jeffrey W. H., Desai, Mahesh N., Finn, Barbara M., Babiarz, Joseph E., Tomaselli, Hollis C.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 552 KB

english, 1985

20

2-Fluoroformycin and 2-aminoformycin. Synthesis and biological activity

Secrist, John A., Shortnacy, Anita T., Montgomery, John A.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 450 KB

english, 1985

21

Masthead

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 151 KB

english, 1985

22

Synthesis and in vitro pharmacology of 7-oxabicyclo[2.2.1]heptane analogs of thromboxane A2/PGH2

Sprague, P. W., Heikes, J. E., Gougoutas, J. Z., Malley, M. F., Harris, D. N., Greenberg, R.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.39 MB

english, 1985

23

Difluorostatine and difluorostatone containing peptides as potent and specific renin inhibitors

Thaisrivongs, Suvit, Pals, Donald T., Kati, Warren M., Turner, Steve R., Thomasco, Lisa M.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 363 KB

english, 1985

24

Antimalarial agents. 1. .alpha.-Santonin-derived cyclic peroxide as potential antimalarial agent

Tani, Shohei, Fukamiya, Narihiko, Kiyokawa, Hiroshi, Musallam, H. A., Pick, Robert O., Lee, Kuo Hsiung

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 282 KB

english, 1985

25

Synthesis and evaluation of potential radioligands for the progesterone receptor

Hoyte, R. M., Rosner, W., Johnson, I. S., Zielinski, J., Hochberg, R. B.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 718 KB

english, 1985

26

Synthesis, characterization, and anorectic testing of the four stereoisomers of cyclo(histidylproline)

Kukla, Michael J., Breslin, Henry J., Bowden, Charles R.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.01 MB

english, 1985

27

Book Reviews

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 312 KB

english, 1985

28

Dog coronary artery adenosine receptor: structure of the N6-alkyl subregion

Kusachi, Shozo, Thompson, Robert D., Bugni, William J., Yamada, Nobuyuki, Olsson, Ray A.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.14 MB

english, 1985

29

Inhibitors of blood platelet aggregation. Effects of some 1,2-benzisothiazol-3-ones on platelet responsiveness to adenosine diphosphate and collagen

Baggaley, Keith H., English, Peter D., Jennings, L. John A., Morgan, Brian, Nunn, Barbara, Tyrrell, A. William R.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 887 KB

english, 1985

30

Alkylating .beta.-blockers: activity of isomeric bromoacetyl alprenolol menthanes

Liptak, Andras, Kusiak, John W., Pitha, Josef

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 753 KB

english, 1985

31

Structure-activity relationships among benextramine-related tetraamine disulfides at peripheral .alpha.-adrenoreceptors

Angeli, Piero, Brasili, Livio, Brancia, Egle, Giardina, Dario, Quaglia, Wilma, Melchiorre, Carlo

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 697 KB

english, 1985

32

Structure-activity relationship studies in the field of calcium(II) antagonists. Effect of modifications at the tetrasubstituted carbon of verapamil-like compounds

Gualtieri, Fulvio, Teodori, Elisabetta, Bellucci, Cristina, Pesce, Edilio, Piacenza, Giuseppe

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.00 MB

english, 1985

33

Evaluation of the brain-specific delivery of radioiodinated (Iodophenyl) alkyl-substituted amines coupled to a dihydropyridine carrier

Tedjamulia, M. L., Srivastava, P. C., Knapp, F. F.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 948 KB

english, 1985

34

Synthesis and pharmacology of the potent angiotensin-converting enzyme inhibitor N-[1(S)-(ethoxycarbonyl)-3-phenylpropyl]-(S)-alanyl-(S)-pyroglutamic acid

Johnson, Alexander L., Price, William A., Wong, Pancras C., Vavala, Robert F., Stump, John M.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.01 MB

english, 1985

35

New bicyclic antidepressant agent. Synthesis and activity of napactadine and related compounds

McCarthy, James R., Wright, Donald L., Schuster, Albert J., Abdallah, Abdul H., Shea, Philip J., Eyster, Randy

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 692 KB

english, 1985

36

Angiotensin converting enzyme inhibitors: N-substituted D-glutamic acid .gamma.-dipeptides

Ksander, Gary M., Yuan, Andrew M., Diefenbacher, Clive G., Stanton, James L.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 897 KB

english, 1985

37

Novel bis[1,6-dihydro-6,6-dimethyl-1,3,5-triazine-2,4-diamines] as antitrypanosomal agents

Turner, William R., Werbel, Leslie M.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 1.12 MB

english, 1985

38

Study on the inhibition of adenosine deaminase

Montgomery, John A., Thomas, H. Jeanette, Zell, Alan L., Einsphar, Howard M., Bugg, Charles E.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 455 KB

english, 1985

39

GABA agonists. Resolution, absolute stereochemistry and enantioselectivity of (S)-(+)- and (R)-(-)-dihydromuscimol

Krogsgaard-Larsen, Povl, Nielsen, Lone, Falch, Erik, Curtis, David R.

Journal:

Journal of Medicinal Chemistry

Year:

1985

Language:

english

File:

PDF, 835 KB

english, 1985

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