Volume 44; Issue 19

Journal of Medicinal Chemistry

Volume 44; Issue 19

1

Design and Synthesis of [(2,3-Dichlorophenyl)piperazin-1-yl]alkylfluorenylcarboxamides as Novel Ligands Selective for the Dopamine D 3 Receptor Subtype

Robarge, Michael J., Husbands, Stephen M., Kieltyka, Andrzej, Brodbeck, Robbin, Thurkauf, Andrew, Newman, Amy Hauck

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 153 KB

english, 2001

2

Synthesis and Evaluation of Cryptolepine Analogues for Their Potential as New Antimalarial Agents

Wright, Colin W., Addae-Kyereme, Jonathan, Breen, Anthony G., Brown, John E., Cox, Marlene F., Croft, Simon L., Gökçek, Yaman, Kendrick, Howard, Phillips, Roger M., Pollet, Pamela L.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 101 KB

english, 2001

3

Coumarins Derivatives as Dual Inhibitors of Acetylcholinesterase and Monoamine Oxidase

Brühlmann, Corinne, Ooms, Frédéric, Carrupt, Pierre-Alain, Testa, Bernard, Catto, Marco, Leonetti, Francesco, Altomare, Cosimo, Carotti, Angelo

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 48 KB

english, 2001

4

Acyclic and Cyclopropyl Analogues of Adenosine Bisphosphate Antagonists of the P2Y 1 Receptor: Structure−Activity Relationships and Receptor Docking

Kim, Hak Sung, Barak, Dov, Harden, T. Kendall, Boyer, José L., Jacobson, Kenneth A.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 566 KB

english, 2001

5

Antimalarial Simplified 3-Aryltrioxanes: Synthesis and Preclinical Efficacy/Toxicity Testing in Rodents

Posner, Gary H., Jeon, Heung Bae, Parker, Michael H., Krasavin, Mikhail, Paik, Ik-Hyeon, Shapiro, Theresa A.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 125 KB

english, 2001

6

Design and Synthesis of Potent C 2 -Symmetric Diol-Based HIV-1 Protease Inhibitors: Effects of Fluoro Substitution

Pyring, David, Lindberg, Jimmy, Rosenquist, Åsa, Zuccarello, Guido, Kvarnström, Ingemar, Zhang, Hong, Vrang, Lotta, Unge, Torsten, Classon, Bjorn, Hallberg, Anders, Samuelsson, Bertil

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 138 KB

english, 2001

7

Fourier Transform Infrared Investigation of Non-Heme Fe(III) and Fe(II) Decomposition of Artemisinin and of a Simplified Trioxane Alcohol

Kapetanaki, Sofia, Varotsis, Constantinos

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 95 KB

english, 2001

8

Synthesis, Ionotropic Glutamate Receptor Binding Affinity, and Structure−Activity Relationships of a New Set of 4,5-Dihydro-8-heteroaryl-4-oxo-1,2,4-triazolo[1,5- a ]quinoxaline-2-carboxylates Analogues of TQX-173

Catarzi, Daniela, Colotta, Vittoria, Varano, Flavia, Filacchioni, Guido, Galli, Alessandro, Costagli, Chiara, Carlà, Vincenzo

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 104 KB

english, 2001

9

Properties and Interaction of Heterologously Expressed Glutamate Decarboxylase Isoenzymes GAD 65kDa and GAD 67kDa from Human Brain with Ginkgotoxin and Its 5‘-Phosphate

Buss, Katrin, Drewke, Christel, Lohmann, Stephanie, Piwonska, Agata, Leistner, Eckhard

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 113 KB

english, 2001

10

[2‘,6‘-Dimethyltyrosine]Dynorphin A(1−11)-NH 2 Analogues Lacking an N-Terminal Amino Group: Potent and Selective κ Opioid Antagonists

Lu, Yixin, Nguyen, Thi M.-D., Weltrowska, Grazyna, Berezowska, Irena, Lemieux, Carole, Chung, Nga N., Schiller, Peter W.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 58 KB

english, 2001

11

Ordered Water and Ligand Mobility in the HIV-1 Integrase-5CITEP Complex: A Molecular Dynamics Study

Ni,, Sotriffer, Christoph A., McCammon, J. Andrew

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 120 KB

english, 2001

12

Identification of Alkylidene Hydrazides as Glucagon Receptor Antagonists

Ling, Anthony, Hong, Yufeng, Gonzalez, Javier, Gregor, Vlad, Polinsky, Alex, Kuki, Atsuo, Shi, Shenghua, Teston, Kimberly, Murphy, Douglas, Porter, John, Kiel, Dan, Lakis, James, Anderes, Kenna, May,

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 115 KB

english, 2001

13

N -Aryl Sulfonyl Homocysteine Hydroxamate Inhibitors of Matrix Metalloproteinases: Further Probing of the S 1 , S 1 ‘, and S 2 ‘ Pockets

Hanessian, Stephen, Moitessier, Nicolas, Gauchet, Cécile, Viau, Martin

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 97 KB

english, 2001

14

A New Approach to Search for the Bioactive Conformation of Glucagon: Positional Cyclization Scanning

Ahn, Jung-Mo, Gitu, Peter M., Medeiros, Matthew, Swift, Jennifer R., Trivedi, Dev, Hruby, Victor J.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 135 KB

english, 2001

15

[ 99m Tc]Oxotechnetium(V) Complexes of Amine-Amide-Dithiol Chelates with Dialkylaminoalkyl Substituents as Potential Diagnostic Probes for Malignant Melanoma

Friebe, Matthias, Mahmood, Ashfaq, Bolzati, Cristina, Drews, Antje, Johannsen, Bernd, Eisenhut, Michael, Kraemer, Daniel, Davison, Alan, Jones, Alun G.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 130 KB

english, 2001

16

Determination of the Binding Specificity of an Integral Membrane Protein by Saturation Transfer Difference NMR: RGD Peptide Ligands Binding to Integrin α IIb β 3†

Meinecke, Robert, Meyer, Bernd

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 182 KB

english, 2001

17

Synthesis and Conformational Analysis of Fusidic Acid Side Chain Derivatives in Relation to Antibacterial Activity

Duvold, Tore, Sørensen, Morten Dahl, Björkling, Fredrik, Henriksen, Anne S., Rastrup-Andersen, Niels

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 144 KB

english, 2001

18

Design and Synthesis of Matrix Metalloproteinase Inhibitors Guided by Molecular Modeling. Picking the S 1 Pocket Using Conformationally Constrained Inhibitors

Hanessian, Stephen, MacKay, D. Bruce, Moitessier, Nicolas

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 285 KB

english, 2001

19

Exploration of Novel Aryl Binding Sites of Farnesyltransferase Using Molecular Modeling and Benzophenone-Based Farnesyltransferase Inhibitors

Böhm, Markus, Mitsch, Andreas, Wissner, Pia, Sattler, Isabel, Schlitzer, Martin

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 1.33 MB

english, 2001

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