Volume 44; Issue 3

Journal of Medicinal Chemistry

Volume 44; Issue 3

1

Synthesis and SAR of a New Series of COX-2-Selective Inhibitors: Pyrazolo[1,5-a]pyrimidines

Almansa, Carmen, de Arriba, Alberto F., Cavalcanti, Fernando L., Gómez, Luis A., Miralles, Agustí, Merlos, Manuel, García-Rafanell, Julián, Forn, Javier

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 191 KB

english, 2001

2

3-Aryl[1,2,4]triazino[4,3-a]benzimidazol-4(10H)-ones: A New Class of Selective A1 Adenosine Receptor Antagonists

Da Settimo, Federico, Primofiore, Giampaolo, Taliani, Sabrina, Marini, Anna Maria, La Motta, Concettina, Novellino, Ettore, Greco, Giovanni, Lavecchia, Antonio, Trincavelli, Letizia, Martini, Claudia

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 560 KB

english, 2001

3

Calculation of the Hydrophobicity of Platinum Drugs

Platts, James A., Hibbs, David E., Hambley, Trevor W., Hall, Matthew D.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 76 KB

english, 2001

4

Quinoxalinylethylpyridylthioureas (QXPTs) as Potent Non-Nucleoside HIV-1 Reverse Transcriptase (RT) Inhibitors. Further SAR Studies and Identification of a Novel Orally Bioavailable Hydrazine-Based Antiviral Agent

Campiani, Giuseppe, Aiello, Francesca, Fabbrini, Monica, Morelli, Elena, Ramunno, Anna, Armaroli, Silvia, Nacci, Vito, Garofalo, Antonio, Greco, Giovanni, Novellino, Ettore, Maga, Giovanni, Spadari, S

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 216 KB

english, 2001

5

GnRH Antagonists: A New Generation of Long Acting Analogues Incorporating p -Ureido-phenylalanines at Positions 5 and 6 †

Jiang, Guangcheng, Stalewski, Jacek, Galyean, Robert, Dykert, John, Schteingart, Claudio, Broqua, Pierre, Aebi, Audrey, Aubert, Michel L., Semple, Graeme, Robson, Peter, Akinsanya, Karen, Haigh, Rober

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 231 KB

english, 2001

6

Behavioral Approach to Nondyskinetic Dopamine Antagonists: Identification of Seroquel

Warawa, Edward J., Migler, Bernard M., Ohnmacht, Cyrus J., Needles, Ann L., Gatos, George C., McLaren, Frances M., Nelson, Cynthia L., Kirkland, Karen M.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 198 KB

english, 2001

7

Cis- Unsaturated Analogues of 3,8,13,18,23-Pentaazapentacosane (BE-4-4-4-4): Synthesis and Growth Inhibitory Effects on Human Prostate Cancer Cell Lines

Reddy, Venodhar K., Sarkar, Aparajita, Valasinas, Aldonia, Marton, Laurence J., Basu, Hirak S., Frydman, Benjamin

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 254 KB

english, 2001

8

Conformationally Restricted Analogues of 1N , 14N -Bisethylhomospermine (BE-4-4-4): Synthesis and Growth Inhibitory Effects on Human Prostate Cancer Cells

Valasinas, Aldonia, Sarkar, Aparajita, Reddy, Venodhar K., Marton, Laurence J., Basu, Hirak S., Frydman, Benjamin

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 283 KB

english, 2001

9

[ 3 H] N -2-(4-( N -Benzamido)phenyl)propyl-2- propanesulfonamide: A Novel AMPA Receptor Potentiator and Radioligand

Zarrinmayeh, Hamideh, Bleakman, David, Gates, Mary R., Yu, Hong, Zimmerman, Dennis M., Ornstein, Paul L., McKennon, Tracey, Arnold, M. Brian, Wheeler, William J., Skolnick, Phil

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 56 KB

english, 2001

10

Tyrosine Kinase Inhibitors. 18. 6-Substituted 4-Anilinoquinazolines and 4-Anilinopyrido[3,4- d ]pyrimidines as Soluble, Irreversible Inhibitors of the Epidermal Growth Factor Receptor

Smaill, Jeff B., Showalter, H. D. Hollis, Zhou, Hairong, Bridges, Alexander J., McNamara, Dennis J., Fry, David W., Nelson, James M., Sherwood, Veronika, Vincent, Patrick W., Roberts, Bill J., Elliott

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 160 KB

english, 2001

11

Analogues of Prazosin That Bear a Benextramine-Related Polyamine Backbone Exhibit Different Antagonism toward α 1 -Adrenoreceptor Subtypes

Bolognesi, Maria L., Marucci, Gabriella, Angeli, Piero, Buccioni, Michela, Minarini, Anna, Rosini, Michela, Tumiatti, Vincenzo, Melchiorre, Carlo

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 130 KB

english, 2001

12

Oral Drug Absorption Prediction and Assessment Edited by Jennifer B. Dressman and Hans Lennermäs. Marcel Dekker, Inc., New York. 2000. x + 330 pp. 16 × 23.5 cm. ISBN 0-8247-0272-7. $165.00.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 15 KB

english, 2001

13

Synthesis by Chemoselective Ligation and Biological Evaluation of Novel Cell-Permeable PKC-ζ Pseudosubstrate Lipopeptides

Bonnet, Dominique, Thiam, Kader, Loing, Estelle, Melnyk, Oleg, Gras-Masse, Hélène

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 66 KB

english, 2001

14

Design, Synthesis, and Modeling of Novel Cyclic Thrombin Receptor-Derived Peptide Analogues of the Ser 42 -Phe-Leu-Leu-Arg 46 Motif Sequence with Fixed Conformations of Pharmacophoric Groups: Importance of a Phe/Arg/NH 2 Cluster for Receptor Activation and Implications in the Design of Nonpeptide Thrombin Receptor Mimetics †

Alexopoulos, Kostas, Panagiotopoulos, Dimitris, Mavromoustakos, Thomas, Fatseas, Panagiotis, Paredes-Carbajal, Maria Christina, Mascher, Dieter, Mihailescu, Stefan, Matsoukas, John

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 390 KB

english, 2001

15

Design, Synthesis, and Biological Evaluation of a Series of Lavendustin A Analogues That Inhibit EGFR and Syk Tyrosine Kinases, as Well as Tubulin Polymerization

Mu, Fanrong, Coffing, Stephanie L., Riese, David J., Geahlen, Robert L., Verdier-Pinard, Pascal, Hamel, Ernest, Johnson, Jill, Cushman, Mark

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 132 KB

english, 2001

16

Seafood and Freshwater Toxins: Pharmacology, Physiology, and Detection Edited by L. M. Botana. Marcel Dekker, New York. 2000. xii + 798 pp. 18.5 × 26 cm. ISBN 0-8247-8956-3. $225.00.

Hieble, J. Paul

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 15 KB

english, 2001

17

Design of Remarkably Simple, Yet Potent Urea-Based Inhibitors of Glutamate Carboxypeptidase II (NAALADase)

Kozikowski, Alan P., Nan, Fajun, Conti, Paola, Zhang, Jiazhong, Ramadan, Epolia, Bzdega, Tomasz, Wroblewska, Barbara, Neale, Joseph H., Pshenichkin, Sergey, Wroblewski, Jarda T.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 44 KB

english, 2001

18

New Dermatological Agents for the Treatment of Psoriasis

Thacher, Scott M., Vasudevan, Jayasree, Tsang, Kwok-Yin, Nagpal, Sunil, Chandraratna, Roshantha A. S.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 182 KB

english, 2001

19

New 1-Aryl-3-(4-arylpiperazin-1-yl)propane Derivatives, with Dual Action at 5-HT 1A Serotonin Receptors and Serotonin Transporter, as a New Class of Antidepressants

Martínez-Esparza, Javier, Oficialdegui, Ana-M., Pérez-Silanes, Silvia, Heras, Begoña, Orús, Lara, Palop, Juan-A., Lasheras, Berta, Roca, Joan, Mourelle, Marisa, Bosch, Ana, Del Castillo, Juan-C., Tord

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 117 KB

english, 2001

20

Structure−Activity Relationships of Pyridoxal Phosphate Derivatives as Potent and Selective Antagonists of P2X 1 Receptors

Kim, Yong-Chul, Brown, Sean G., Harden, T. Kendall, Boyer, José L., Dubyak, George, King, Brian F., Burnstock, Geoffrey, Jacobson, Kenneth A.

Journal:

Journal of Medicinal Chemistry

Year:

2001

Language:

english

File:

PDF, 182 KB

english, 2001

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