Volume 59; Issue 25

Journal of Organic Chemistry

Volume 59; Issue 25

1

The Chemistry of Phosphapeptides: Formation of Functionalized Phosphonochloridates under Mild Conditions and Their Reaction with Alcohols and Amines

Malachowski, William P., Coward, James K.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.02 MB

english, 1994

2

Design and Synthesis of a Conformationally Restricted Cysteine Protease Inhibitor

Cheng, Hengmiao, Keitz, Paul, Jones, J. Bryan

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 760 KB

english, 1994

3

Urea-Derivatized p-tert-Butylcalix[4]arenes: Neutral Ligands for Selective Anion Complexation

Scheerder, Jurgen, Fochi, Mariacristina, Engbersen, Johan F. J., Reinhoudt, David N.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.41 MB

english, 1994

4

Synthesis and Exchange Reactions of 1,4,8,11-Tetraazacyclotetradeca-7(E),14(E)-diene-5,12-diones

Hegedus, Louis S., Moser, William H.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 893 KB

english, 1994

5

Boranes in Synthesis. 6. A New Synthesis of .beta.-Amino Alcohols from Epoxides. Use of Lithium Amides and Aminoborane Catalysts To Synthesize .beta.-Amino Alcohols from Terminal and Internal Epoxides in High Yield

Harris, Clifford E., Fisher, Gary B., Beardsley, David, Lee, Lawrence, Goralski, Christian T., Nicholson, Lawrence W., Singaram, Bakthan

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 701 KB

english, 1994

6

On the Stereoselectivity of the Reaction of N-(9-Phenylfluoren-9-yl)aspartate Enolates with Electrophiles. Synthesis of Enantiomerically Pure 3-Hydroxy-, 3-Amino-, and 3-Hydroxy-3-methylaspartates

Fernandez-Megia, Eduardo, Paz, Manuel M., Sardina, F. Javier

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.38 MB

english, 1994

7

Enediyne- and Tributyltin Hydride-Mediated Aryl Radical Additions onto Various Radical Acceptors

Grissom, Janet Wisniewski, Klingberg, Detlef, Meyenburg, Sabine, Stallman, Brenda L.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.71 MB

english, 1994

8

A TMM Cycloaddition Strategy to the Bicyclo[6.3.0]undecyl Ring System. A Total Synthesis of 11-Hydroxyjasionone

Trost, Barry M., Parquette, Jon R.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 242 KB

english, 1994

9

Nonionic Superbase-Promoted Synthesis of Oxazoles and Pyrroles: Facile Synthesis of Porphyrins and .alpha.-C-Acyl Amino Acid Esters

Tang, Jiansheng, Verkade, John G.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.23 MB

english, 1994

10

A New Access to Kainoids via a Tandem Aza-Cope/Mannich Reaction. Application to the Enantioselective Synthesis of (-)-.alpha.-Allokainic Acid

Agami, Claude, Cases, Manuel, Couty, Francois

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 570 KB

english, 1994

11

Syntheses of Strychnos- and Aspidospermatan-Type Alkaloids. 6. Total Syntheses of (.+-.)-Echitamidine, (.+-.)-Alstogustine, (.+-.)-19-epi-Alstogustine, and (.+-.)-Akuammicine

Kuehne, Martin E., Xu, Feng, Brook, Christopher S.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 554 KB

english, 1994

12

Effects of Olefin Geometry on the Stereochemistry of Lewis Acid Mediated Additions of Crotylstannanes to Aldehydes

Keck, Gary E., Savin, Kenneth A., Cressman, Erik N. K., Abbott, Duane E.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.69 MB

english, 1994

13

Syntheses of 4''-epi-Amino-4''-deoxyavermectins B1

Cvetovich, Raymond J., Kelly, Dennis H., DiMichele, Lisa M., Shuman, Richard F., Grabowski, Edward J. J.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 720 KB

english, 1994

14

Practical Synthesis of Chiral Synthons for the Preparation of HMG-CoA Reductase Inhibitors

Konoike, Toshiro, Araki, Yoshitaka

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 815 KB

english, 1994

15

Peroxometalate Catalyzed Oxidations with Hydrogen Peroxide in Biphasic Reaction Media: Reactions in Inverse Emulsions

Neumann, Ronny, Khenkin, Alexander M.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 319 KB

english, 1994

16

Enantioselective Synthesis of Homoallylic Amines by Addition of Allylmetal Reagents to Imines Derived from (S)-Valine Esters

Basile, Tiziana, Bocoum, Allaye, Savoia, Diego, Umani-Ronchi, Achille

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.12 MB

english, 1994

17

Resolution of Amino Acids in a Mixture of 2-Methyl-2-propanol/water (19:1) Catalyzed by Alcalase via in Situ Racemization of One Antipode Mediated by Pyridoxal 5-Phosphate

Chen, Shui-Tein, Huang, Wen-Hong, Wang, Kung-Tsung

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 263 KB

english, 1994

18

Synthesis of New Tetrafluorobenzo Heteroaromatic Compounds

Dolbier, William R., Burkholder, Conrad, Abboud, Khalil A., Loehle, David

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 923 KB

english, 1994

19

Asymmetric Synthesis of Chiral Secondary Alcohols with Isopropyl Substituents by the Catalytic Enantioselective Addition of Diisopropylzinc to Aldehydes using N,N-Dialkylnorephedrines as Chiral Catalysts

Soai, Kenso, Hayase, Tadakatsu, Takai, Kazuhisa, Sugiyama, Tadashi

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 256 KB

english, 1994

20

Thiol Mediated Free Radical Cyclization of Alkenyl and Alkynyl Isocyanides

Bachi, Mario D., Balanov, Anna, Bar-Ner, Nira

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 925 KB

english, 1994

21

Glycosidation Route to 4''-epi-(Methylamino)-4''-Deoxyavermectin B1 (MK-244, Emamectin Benzoate)

Loewe, Mallory F., Cvetovich, Raymond J., DiMichele, Lisa M., Shuman, Richard F., Grabowski, Edward J. J.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 825 KB

english, 1994

22

Stereocontrolled Total Synthesis of Calcitriol Derivatives: 1,25-Dihydroxy-2-(4'-hydroxybutyl)vitamin D3 Analogs of an Osteoporosis Drug

Posner, Gary H., Johnson, Neil

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 848 KB

english, 1994

23

Asymmetric Synthesis of 6,6'-Dialkoxy-2,2'-biphenyldiols by Using Menthone as a Chiral Template

Harada, Toshiro, Ueda, Shinji, Yoshida, Tetsuya, Inoue, Atsushi, Takeuchi, Masahiro, Ogawa, Nobuhiro, Oku, Akira, Shiro, Motoo

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 278 KB

english, 1994

24

Consequences of .alpha.-Bromo Substitution on the Course of Allylmetal Additions to 1-Oxaspiro[4.5]dec-7-en-6-one

Klemeyer, Horst Jan, Paquette, Leo A.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 429 KB

english, 1994

25

Ester Cleavage by Cyclodextrins in Aqueous Dimethyl Sulfoxide Mixtures. Substrate Binding versus Transition State Binding

Tee, Oswald S., Mazza, Charles, Lozano-Hemmer, Rafael, Giorgi, Javier B.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 917 KB

english, 1994

26

Total Synthesis of (.+-.)-Aspidofractinine and (.+-.)-Aspidospermidine

Wenkert, Ernest, Liu, Song

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 791 KB

english, 1994

27

Synthesis and Structure of 2,2'-Dihydroxybenzophenones and 1,8-Dihydroxyfluorenones

Sharma, Vijay, Bachand, Benoit, Simard, Michel, Wuest, James D.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.17 MB

english, 1994

28

Synthesis of [1.1.1.1]Metacyclophane Macrocycle

Rajca, Andrzej, Padmakumar, Raghavakaimal, Smithhisler, Donald J., Desai, Shailesh R., Ross, Charles R., Stezowski, John J.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 447 KB

english, 1994

29

Can Remote Substituent Effects Influence Reactivity and Stereoselectivity in the Diels-Alder Cycloadditions of p-Substituted 6-Phenyl-6-methylfulvenes?

Gugelchuk, M. M., Chan, P. C.-M., Sprules, T. J.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.89 MB

english, 1994

30

Stereospecific Synthesis and NMR Conformational Studies of .gamma.-Butyrolactones of Nucleosides as Chiral Synthons for the Preparation of 2'-C- and 3'-C-Branched-Chain Nucleosides

Velazquez, Sonsoles, Jimeno, Maria Luisa, Huss, Sophie, Balzarini, Jan, Camarasa, Maria-Jose

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.20 MB

english, 1994

31

Silylcarbobicyclization of 1,6-Diynes: A Novel Catalytic Route to Bicyclo[3.3.0]octenones

Ojima, Iwao, Fracchiolla, Dora A., Donovan, Robert J., Banerji, Pratip

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 288 KB

english, 1994

32

3-(Tri-n-butylstannyl)-2-cyclobuten-1-one: Synthesis and Stille Cross-Coupling as a Route to 3-Substituted Cyclobutenones

Liebeskind, Lanny S., Stone, Guy B., Zhang, Shijie

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 494 KB

english, 1994

33

Methods for Combinatorial Organic Synthesis: The Use of Fast 13C NMR Analysis for Gel Phase Reaction Monitoring

Look, Gary C., Holmes, Christopher P., Chinn, Jason P., Gallop, Mark A.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 722 KB

english, 1994

34

Theoretical Characterization of Cycloaddition Reactions of the Cyclopropylcarbinyl Cation

Cramer, Christopher J., Barrows, Susan E.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 555 KB

english, 1994

35

Lewis Acid Promoted Additions of .gamma.-Alkoxy- and -(Silyloxy)crotylstannanes to (S)-2-(Benzyloxy)propanal

Marshall, James A., Jablonowski, Jill A., Luke, George P.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 915 KB

english, 1994

36

Reactions of Benzaldehyde with Thiazolium Salts in Me2SO: Evidence for Initial Formation of 2-(.alpha.-Hydroxybenzyl)thiazolium by Nucleophilic Addition, and for Dramatic Solvent Effects on Benzoin Formation

Chen, Yao-Tsung, Barletta, Gabriel L., Haghjoo, Khadijah, Cheng, Jung Tsang, Jordan, Frank

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.02 MB

english, 1994

37

Stereocontrolled Formation of Quaternary Carbon Centers by Conjugate Addition of Lithium Enolates of Dioxanones to .beta.-Bromoacrylates and .beta.-Bromovinyl Sulfones: Dependence of Stereoselectivity on Alkene Geometry

Bruncko, Milan, Crich, David

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 437 KB

english, 1994

38

Iminodithiocarbonates as Formaldehyde Imine Equivalents: Sequential Two Step Approach to 4-Unsubstituted .beta.-Lactams through Chromium(0) Carbene Photocycloaddition-Nickel Boride Desulfurization

Alcaide, Benito, Casarrubios, Luis, Dominguez, Gema, Sierra, Miguel A.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 439 KB

english, 1994

39

Preparation of 2,2-Dichloro-3(2H)-furanone and Its Reactions with Heteronucleophiles

Murakami, Masahiro, Hayashi, Minoru, Ito, Yoshihiko

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 613 KB

english, 1994

40

General Enantiospecific Route to Isochromanquinones. Synthesis of (-)-Nanaomycin D

Winters, Michael P., Stranberg, Michael, Moore, Harold W.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 268 KB

english, 1994

41

Stannylformylation of 1,6-Dienes Accompanied by Five-Membered Radical Ring Closure

Ryu, Ilhyong, Kurihara, Akio, Muraoka, Hideo, Tsunoi, Shinji, Kambe, Nobuaki, Sonoda, Noboru

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 285 KB

english, 1994

42

Synthesis and Evaluation of 3-Dehydroquinate Synthase Transition State Analogs

Montchamp, Jean-Luc, Frost, J. W.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 780 KB

english, 1994

43

The Chemistry of Phosphapeptides: Investigations on the Synthesis of Phosphonamidate, Phosphonate, and Phosphinate Analogs of Glutamyl-.gamma.-glutamate

Malachowski, William P., Coward, James K.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.08 MB

english, 1994

44

Conformationally Rigid Tricyclic Tripods: Synthesis and Application to Preparation of Enterobactin Analogs

Tse, Bruno, Kishi, Yoshito

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.48 MB

english, 1994

45

On the Transition State of the Chorismate-Prephenate Rearrangement

Wiest, Olaf, Houk, K. N.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.28 MB

english, 1994

46

In Quest of Tricyclo[4.4.1.04,11]undeca-1,3,5,7,9-pentaene, a Highly Strained, Cyclic 10.pi.-Electron, Polyunsaturated Hydrocarbon. Synthesis of a Methoxyl-Substituted Dihydro Derivative

Branan, Bruce M., Paquette, Leo A.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 666 KB

english, 1994

47

Stereoselective Synthesis of .beta.-Oxygenated .alpha.-Hydroxyphosphonates by Lewis Acid-Mediated Stereoselective Hydrophosphonylation of .alpha.-Benzyloxy Aldehydes. An Application to the Synthesis of Phosphonic Acid Analogs of Oxyamino Acids

Yokomatsu, Tsutomu, Yoshida, Yoshinori, Shibuya, Shiroshi

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 481 KB

english, 1994

48

Total Synthesis of ACRL Toxin IIIb: A Protocol for Parlaying Aldols into Synthons Containing Three Stereocenters Having an [n, n + 1, n + 4] Relationship

Munchhof, Michael J., Heathcock, Clayton H.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 221 KB

english, 1994

49

Radical Cations of Benzo[a]pyrene and 6-Substituted Derivatives: Synthesis and Reaction with Nucleophiles

Cremonesi, Paolo, Stack, Douglas E., Rogan, Eleanor G., Cavalieri, Ercole L.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 672 KB

english, 1994

50

Theoretical Study of Ethylene and Vinyl Alcohol Addition to 1,4-Dioxa-1,3-butadiene

Jursic, Branko S., Zdravkovski, Zoran

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 576 KB

english, 1994

51

Kinetic Resolution of Phosphines and Phosphine Oxides with Phosphorus Stereocenters by Hydrolases

Serreqi, Alessio N., Kazlauskas, Romas J.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 975 KB

english, 1994

52

Synthesis of .alpha.-Pyridone-Based Azaheteroaromatics by Intramolecular Vinylketene Cyclizations onto the C:N Bond of Nitrogen Heteroaromatics

Birchler, Angela Gurski, Liu, Fuqiang, Liebeskind, Lanny S.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.20 MB

english, 1994

53

Remote Conformational Bias Effects on Diastereofacial Selectivity in SE2' Additions of .gamma.-Oxygenated Allylic Stannanes to Chiral Enals

Marshall, James A., Beaudoin, Serge

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 763 KB

english, 1994

54

Stereoselective Synthesis of 2'-Deoxy-.beta.-D-threo-pentofuranosyl Nucleosides by the NBS-Promoted Coupling Reaction of Thioglycosides with Silylated Heterocyclic Bases

Sugimura, Hideyuki, Osumi, Kenji, Kodaka, Yasuko, Sujino, Keiko

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.07 MB

english, 1994

55

Diastereoselective .alpha.-Alkylation of 2-Acyl-3-phenyl-l-menthopyrazoles

Kashima, Choji, Fukuchi, Iwao, Hosomi, Akira

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 493 KB

english, 1994

56

A Novel, Mild, and Practical Regeneration of Alcohols from their Allylic Ethers by NBS/H2O

Robles Diaz, Rafael, Rodriguez Melgarejo, Concepcion, Plaza Lopez-Espinosa, Maria T., Izquierdo Cubero, Isidoro

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 238 KB

english, 1994

57

Stereoselective Synthesis of 6-Substituted Decahydroisoquinoline-3-carboxylates: Intermediates for the Preparation of Conformationally Constrained Acidic Amino Acids

Ornstein, Paul L., Augenstein, Nancy K., Arnold, M. Brian

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1018 KB

english, 1994

58

Editorial

Heathcock, Clayton

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 75 KB

english, 1994

59

Rearrangement of (Polymethoxybenzyl)ammonium N-Methylides

Maeda, Yasuhiro, Shirai, Naohiro, Sato, Yoshiro, Tatewaki, Hiroshi

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 631 KB

english, 1994

60

Synthesis, Characterization, and Alkali Metal Stability Constants of a New Bis(phosphotriester) Macrobicyclic Polyether Cryptand

Allan, Christian B., Spreer, Larry O.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 746 KB

english, 1994

61

Ruthenium Complex-Catalyzed Carbonylation of Allylic Compounds

Mitsudo, Take-aki, Suzuki, Nobuyoshi, Kondo, Teruyuki, Watanabe, Yoshihisa

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 808 KB

english, 1994

62

New Generation Method for a Samarium(II) Equivalent: Me3SiX (X = Br and I)/Sm-Assisted Intermolecular Carbon-Carbon Bond Forming Reactions of Carbonyl Compounds

Akane, Noriyuki, Hatano, Tadashi, Kusui, Hiroko, Nishiyama, Yutaka, Ishii, Yasutaka

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 707 KB

english, 1994

63

Asymmetric Diels-Alder Reactions of Chiral (E)-2-Cyanocinnamates. 2. Synthesis of the Four 1-Amino-2-phenyl-1-cyclohexanecarboxylic Acids in Enantiomerically Pure Form

Cativiela, Carlos, Avenoza, Alberto, Paris, Miguel, Peregrina, Jesus M.

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 707 KB

english, 1994

64

A Novel Synthesis of Methyl 1,5-Disubstituted Imidazole-4-carboxylates Using 3-Bromo-2-isocyanoacrylates (BICA)

Nunami, Ken-ichi, Yamada, Masaki, Fukui, Toshio, Matsumoto, Kazuo

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.01 MB

english, 1994

65

Dualistic Reactivity of Lithium and Zinc Dienolates with Imines: Effects of Counterion, Temperature, and Substituents on .alpha.- and .gamma.-Coupling

van Maanen, Hendrik L., Kleijn, Henk, Jastrzebski, Johann T. B. H., Lakin, Miles T., Spek, Anthony L., van Koten, Gerard

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 1.68 MB

english, 1994

66

New 1H and 13C NMR Spectral Data on "Higher Order" Cyanocuprates. If the Cyano Ligand Is Not On Copper, Then Where Is It?

Lipshutz, Bruce H., James, Brian

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 739 KB

english, 1994

67

Masthead

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 164 KB

english, 1994

68

Novel Cyclopentenone Synthesis by Base-Catalyzed Cyclization of Dienediones

Ong, Chi Wi, Chen, Chong Ming, Juang, Shyh Shian

Journal:

Journal of Organic Chemistry

Year:

1994

Language:

english

File:

PDF, 239 KB

english, 1994