Volume 2; Issue 9

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MedChemComm
Volume 2; Issue 9

MedChemComm

Volume 2; Issue 9

1

Identification of CYP1A2 ligands by structure-based and ligand-based virtual screening

Lastdrager, Jeroen, Oostenbrink, Chris, Vasanthanathan, Poongavanam, Commandeur, Jan N. M., Vermeulen, Nico P. E., Jørgensen, Flemming S., Olsen, Lars

Journal:

Year:

2011

Language:

english

File:

PDF, 517 KB

english, 2011

2

Synthesis and biological evaluation of 2,3-bis(het)aryl-4-azaindole derivatives as protein kinase inhibitors

Pin, Frédéric, Buron, Frédéric, Saab, Fabienne, Colliandre, Lionel, Bourg, Stéphane, Schoentgen, Françoise, Le Guevel, Remy, Guillouzo, Christiane, Routier, Sylvain

Journal:

Year:

2011

Language:

english

File:

PDF, 230 KB

english, 2011

3

Chemometric modeling and pharmacophore mapping in coronary heart disease: 2-arylbenzoxazoles as cholesteryl ester transfer protein inhibitors

Jana, Dhritiman, Halder, Amit Kumar, Adhikari, Nilanjan, Maiti, Milan Kumar, Mondal, Chanchal, Jha, Tarun

Journal:

Year:

2011

Language:

english

File:

PDF, 518 KB

english, 2011

4

2-Anilinonicotinyl linked 1,3,4-oxadiazole derivatives: Synthesis, antitumour activity and inhibition of tubulin polymerization

Kamal, Ahmed, Srikanth, Y. V. V., Shaik, Thokhir B., Khan, M. Naseer A., Ashraf, Md., Reddy, M. Kashi, Kumar, K. Anil, Kalivendi, Shasi V.

Journal:

Year:

2011

Language:

english

File:

PDF, 28.06 MB

english, 2011

5

Designing glucokinase activators with reduced hypoglycemia risk: discovery of N,N-dimethyl-5-(2-methyl-6-((5-methylpyrazin-2-yl)-carbamoyl)benzofuran-4-yloxy)pyrimidine-2-carboxamide as a clinical candidate for the treatment of type 2 diabetes mellitus

Pfefferkorn, Jeffrey A., Guzman-Perez, Angel, Oates, Peter J., Litchfield, John, Aspnes, Gary, Basak, Arindrajit, Benbow, John, Berliner, Martin A., Bian, Jianwei, Choi, Chulho, Freeman-Cook, Kevin, C

Journal:

Year:

2011

Language:

english

File:

PDF, 652 KB

english, 2011

6

p-Carborane-based androgen antagonists active in LNCaP cells with a mutated androgen receptor

Fujii, Shinya, Yamada, Ayumi, Tomita, Keiko, Nagano, Mao, Goto, Tokuhito, Ohta, Kiminori, Harayama, Takashi, Endo, Yasuyuki, Kagechika, Hiroyuki

Journal:

Year:

2011

Language:

english

File:

PDF, 112 KB

english, 2011

7

20-O-IngenolEZ, a catalytic topoisomerase II inhibitor, specifically inhibits cell proliferation and induces double-strand DNA breaks in BLM-/- cells

Watanabe, Manami, Kamada, Yuta, Miyazaki, Khosuke, Mizoguchi, Shoko, Matsuzaki, Keiichi, Kitanaka, Susumu, Miyata, Shohei

Journal:

Year:

2011

Language:

english

File:

PDF, 169 KB

english, 2011

8

Design, synthesis, and structure–activity relationships of 1,3,4-oxadiazol-2(3H)-ones as novel FAAH inhibitors

Kiss, László E., Ferreira, Humberto S., Beliaev, Alexandre, Torrão, Leonel, Bonifácio, Maria João, Learmonth, David A.

Journal:

Year:

2011

Language:

english

File:

PDF, 137 KB

english, 2011

9

Back cover

Journal:

Year:

2011

Language:

english

File:

PDF, 714 KB

english, 2011

10

Pharmacological properties of indolone-N-oxides controlled by a bioreductive transformation in red blood cells?

Ibrahim, Hany, Pantaleo, Antonella, Turrini, Francesco, Arese, Paolo, Nallet, Jean-Pierre, Nepveu, Françoise

Journal:

Year:

2011

Language:

english

File:

PDF, 433 KB

english, 2011

11

Modular assembly of cytotoxic acetogenin mimetics by click linkage with nitrogen functionalities

Mao, Chan, Han, Bing, Wang, Li-Shun, Wang, Shaozhong, Yao, Zhu-Jun

Journal:

Year:

2011

Language:

english

File:

PDF, 318 KB

english, 2011

12

Design and syntheses of some iminosugar derivatives as potential immunosuppressants

Zhang, Guo-Liang, Zheng, Xiu-Jing, Zhang, Li-He, Ye, Xin-Shan

Journal:

Year:

2011

Language:

english

File:

PDF, 240 KB

english, 2011

13

Design, synthesis and initial biological evaluation of a novel pladienolide analog scaffold

Gundluru, Mahesh Kumar, Pourpak, Alan, Cui, Xiaoli, Morris, Stephan W., Webb, Thomas R.

Journal:

Year:

2011

Language:

english

File:

PDF, 203 KB

english, 2011

14

A novel strategy for the synthesis of enzymatically stable biotin–DOTA conjugates for in vivo use

Turhanen, Petri A., Weisell, Janne, Lehtolainen-Dalkilic, Pauliina, Määttä, Ann-Marie, Vepsäläinen, Jouko, Närvänen, Ale

Journal:

Year:

2011

Language:

english

File:

PDF, 90 KB

english, 2011

15

Optimized glucuronidation of dual pharmacology β-2 agonists/M3 antagonists for the treatment of COPD

Hilton, Laura, Osborne, Rachel, Kenyon, Amy S., Baldock, Helen, Bunnage, Mark E., Burrows, Jane, Clarke, Nick, Coghlan, Michele, Entwistle, David, Fairman, David, Feeder, Neil, James, Kim, Jones, Rhys

Journal:

Year:

2011

Language:

english

File:

PDF, 277 KB

english, 2011

16

Enantioselective preparation of ferrocenyl amino phosphines and their cytotoxic activities

Kok, Stanton Hon-lung, Lam, Wing-sze, Chan, Albert Sun-chi, Wong, Wai-yeung, Gambari, Roberto, Wong, Raymond Siu-ming, Lee, Kenneth Ka-ho, Tang, Johnny Cheuk-on, Lam, Kim-hung, Chui, Chung-hin

Journal:

Year:

2011

Language:

english

File:

PDF, 199 KB

english, 2011

17

Front cover

Journal:

Year:

2011

Language:

english

File:

PDF, 714 KB

english, 2011

18

N-Substituted salicylamides as selective malaria parasite dihydroorotate dehydrogenase inhibitors

Fritzson, Ingela, Bedingfield, Paul T. P., Sundin, Anders P., McConkey, Glenn, Nilsson, Ulf J.

Journal:

Year:

2011

Language:

english

File:

PDF, 124 KB

english, 2011

19

Contents list

Journal:

Year:

2011

Language:

english

File:

PDF, 2.39 MB

english, 2011

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