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Volume 22; Issue 2
Main
Medicinal Chemistry Research
Volume 22; Issue 2
Medicinal Chemistry Research
Volume 22; Issue 2
1
Synthesis, characterization, anticancer, and antioxidant activity of some new thiazolidin-4-ones in MCF-7 cells
Arun M. Isloor, Dhanya Sunil, Prakash Shetty, Shridhar Malladi, K. S. R. Pai, Naseer Maliyakkl
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 491 KB
Your tags:
english, 2013
2
A comprehensive structure–activity analysis 2,3,5-trisubstituted 4,5-dihydro-4-oxo-3H-imidazo [4,5-c] pyridine derivatives as angiotensin II receptor antagonists: using 2D- and 3D-QSAR approach
Mukesh C. Sharma, D. V. Kohli
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 974 KB
Your tags:
english, 2013
3
Synthesis and in vitro antibacterial activity of schiff bases ofN-substituted isatins as effective scaffolds
Garima Kumari, Ramendra K. Singh
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 341 KB
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english, 2013
4
Synthesis and antimicrobial activity of coumarin pyrazole pyrimidine 2,4,6(1H,3H,5H)triones and thioxopyrimidine4,6(1H,5H)diones
S. Vijaya Laxmi, B. Suresh Kuarm, B. Rajitha
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 257 KB
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english, 2013
5
Atom-based 3D QSAR studies on novelN-β-d-xylosylindole derivatives as SGLT2 inhibitors
Venkatesan Suryanarayanan, Arumugam Sudha, Sundararaj Rajamanikandan, Ramar Vanajothi, Pappu Srinivasan
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 473 KB
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english, 2013
6
Binding site analysis, 3D-QSAR studies, and molecular design of flavonoids derivatives as potent neuraminidase inhibitors
Jiaying Sun, Hu Mei
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 1009 KB
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english, 2013
7
In vitro antimicrobial and antimycobacterial activity of some chalcones and their derivatives
Divyesh Patel, Premlata Kumari, Navin B. Patel
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 421 KB
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english, 2013
8
Pyrazolo[3,4-d]pyrimidine analogues: synthesis, characterization and their in vitro antiamoebic activity
Shadab Miyan Siddiqui, Attar Salahuddin, Amir Azam
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 762 KB
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english, 2013
9
Quinoline-based azetidinone and thiazolidinone analogues as antimicrobial and antituberculosis agents
Bhupendra M. Mistry, Smita Jauhari
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 415 KB
Your tags:
english, 2013
10
Synthesis, structure, and biological assay of cinnamic amides as potential EGFR kinase inhibitors
Mao Zhang, Xiang Lu, Hong-Jia Zhang, Na Li, Yu Xiao, Hai-Liang Zhu, Yong-Hao Ye
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 390 KB
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english, 2013
11
Spectroscopic characterization of noveld-amino acid-Schiff bases and their Cr(III) and Ni(II) complexes as antimicrobial agents
Nurşen Sarı, Nihat Pişkin, Hatice Öğütcü, Nurdan Kurnaz
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 419 KB
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english, 2013
12
Synthesis and evaluation of analgesic, anti-inflammatory, and anticancer activities of new pyrazole-3(5)-carboxylic acid derivatives
Burcu Çalışkan, Akın Yılmaz, İlker Evren, Sevda Menevşe, Orhan Uludag, Erden Banoglu
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 384 KB
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english, 2013
13
Discovery of novel DPP IV inhibitors: application of pharmacophore-based virtual screening
Jyoti Sharma, Divya Yadav, Sarvesh Paliwal
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 1.01 MB
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english, 2013
14
Immunomodulatory active steroidal saponins fromAsparagus racemosus
Upendra Sharma, Neeraj Kumar, Bikram Singh, Renuka K. Munshi, Supriya Bhalerao
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 264 KB
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english, 2013
15
In vitro antiproliferative effect of β-phenylethylamine derivatives and doxorubicin combinations on MCF/ADR cell lines
Wanda P. Almeida, Paula C. Huber, Luciana K. Kohn, João E. de Carvalho
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 377 KB
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english, 2013
16
Novel 2-thiopyrimidine derivatives as CDK2 inhibitors: molecular modeling, synthesis, and anti-tumor activity evaluation
Omar Abd El-Fattah M. Fathalla, Mohamed A. H. Ismail, Manal M. Anwar, Khaled A. M. Abouzid, Aisha A. K. Ramadan
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 783 KB
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english, 2013
17
Synthesis and biological evaluation of gallic acid analogs
Maurizio Barontini, Ilaria Proietti Silvestri, Valentina Nardi, Fernanda Crisante, Gaetano Pepe, Luigi Pari, Francesco Gallucci, Paolo Bovicelli, Giuliana Righi
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 504 KB
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english, 2013
18
Action of benzimidazolo-piperazinyl derivatives on dopamine receptors
Zenish J. Jain, Rani S. Kankate, Bhavinkumar N. Chaudhari, Rohini D. Kakad
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 574 KB
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english, 2013
19
From peptides to peptidomimetics: rational design of potential PKC-β II inhibitors
P. Sri Divya, Kapil Jain, M. Elizabeth Sobhia
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 519 KB
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english, 2013
20
Design, synthesis, and biological evaluation of new 4-thiazolidinone derivatives substituted with benzimidazole ring as potential chemotherapeutic agents
Georgina N. Masoud, Amal M. Youssef, Magdy M. Abdel Khalek, Abeer E. Abdel Wahab, Ibrahim M. Labouta, Aly A. B. Hazzaa
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 863 KB
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english, 2013
21
Synthesis, structure, and estrogenic activity of 2- and 3-substituted 2,3-dihydro-4H-1-benzopyran-4-ones
Yves Jacquot, Cillian Byrne, Alain Xicluna, Guy Leclercq
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 580 KB
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english, 2013
22
Synthesis of imidazole-derived steroidal hybrids as potent aromatase inhibitors
Ranju Bansal, Sheetal Guleria, Sridhar Thota, Rolf W. Hartmann, Christina Zimmer
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 328 KB
Your tags:
english, 2013
23
Synthesis and in vitro antimicrobial and anti-tubercular evaluation of some quinoline-based azitidinone and thiazolidinone analogues
Bhupendra M. Mistry, Smita Jauhari
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 314 KB
Your tags:
english, 2013
24
Synthesis and antioxidant studies of novelN-substituted benzyl/phenyl-2-(3,4-dimethyl-5,5-dioxidopyrazolo[4,3-c][1,2]benzothiazin-2(4H)-yl)acetamides
Matloob Ahmad, Hamid Latif Siddiqui, John M. Gardiner, Masood Parvez, Sana Aslam
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 428 KB
Your tags:
english, 2013
25
Synthesis and antimicrobial screening of 4-thiazolidinone and 2-azetidinone derivatives of piperazine
Sunil G. Shingade, Sanjaykumar B. Bari
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 268 KB
Your tags:
english, 2013
26
Identification of an antiepileptic lead compound with a more selective activity and its analogues for GABA-AT using in silico approach
Hina Naz Khan, Saima Kulsoom, Hamid Rashid
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 884 KB
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english, 2013
27
Synthesis of newN-arylamino(2-furyl)methylphosphonic acid diesters, and in vitro evaluation of their cytotoxicity against esophageal cancer cells
Anna Agnieszka Klimczak, Agnieszka Kuropatwa, Jarosław Lewkowski, Janusz Szemraj
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 529 KB
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english, 2013
28
Synthesis, antimicrobial and antioxidant activities of some new indole derivatives containing pyridopyrimidine and pyrazolopyridine moieties
Anand R. Saundane, Katkar Vijaykumar, A. V. Vaijinath, Prabhaker Walmik
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 509 KB
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english, 2013
29
Analysis of 6-methoxy podophyllotoxin and podophyllotoxin in hairy root cultures ofLinum albumKotschy ex Boiss
Najmeh Ahmadian Chashmi, Mozafar Sharifi, Morteza Yousefzadi, Mehrdad Behmanesh, Hassan Rezadoost, Alejandra Cardillo, Javier Palazon
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 419 KB
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english, 2013
30
Anti-inflammatory and selective COX-2 inhibitory activities of metal complexes of Schiff bases derived from aldoses
Mohammad S. Iqbal, Syed J. Khurshid, Bakhtiar Muhammad
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 293 KB
Your tags:
english, 2013
31
Synthesis and evaluation of antioxidant activity of 2-styrylchromones
Shrinivas P. Pawar, Dasharath D. Kondhare, P. K. Zubaidha
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 272 KB
Your tags:
english, 2013
32
Synthesis and antibacterial, antimycobacterial and docking studies of novelN-piperazinyl fluoroquinolones
Kapil M. Agrawal, Gokul S. Talele
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 473 KB
Your tags:
english, 2013
33
Essential oil composition, insecticidal and antibacterial activities ofSalvia tomentosaMiller
Zeynep Ulukanli, Salih Karabörklü, Menderes Cenet, Osman Sagdic, Ismet Ozturk, Mehmet Balcilar
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 326 KB
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english, 2013
34
Synthesis and biological evaluation of novel benzoquinones as potential antimicrobial agents
Ibrahim Chaaban, El Sayeda M. El Khawass, Mona A. Mahran, Heba A. Abd El Razik, Nehad S. El Salamouni, Abeer E. Abdel Wahab
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 332 KB
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english, 2013
35
Colchicine and its various physicochemical and biological aspects
Sameer Sapra, Yashika Bhalla, Nandani, Sahil Sharma, Gagandip Singh, Kunal Nepali, Abhishek Budhiraja, Kanaya L. Dhar
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 689 KB
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english, 2013
36
Novel quinazolinone derivatives: synthesis and antimicrobial activity
Osman M. O. Habib, Hussein M. Hassan, Ahmed El-Mekabaty
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 553 KB
Your tags:
english, 2013
37
Synthesis and evaluation of antibacterial and antitubercular activities of some novel imidazo[2,1-b][1,3,4]thiadiazole derivatives
S. D. Joshi, K. Manish, Aravind Badiger
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 320 KB
Your tags:
english, 2013
38
QSAR and pharmacophore modeling ofN-acetyl-2-aminobenzothiazole class of phosphoinositide-3-kinase-α inhibitors
Sandip B. Bharate, Baljinder Singh, Jaideep B. Bharate, Shreyans K. Jain, Samdarshi Meena, Ram A. Vishwakarma
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 710 KB
Your tags:
english, 2013
39
In silico ligand-based pharmacophore model generation for the identification of novelPneumocystis cariniiDHFR inhibitors
Yusra Sajid Kiani, Saima Kalsoom, Naveeda Riaz
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 1.99 MB
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english, 2013
40
Synthesis of novel benzimidazole derivatives: as potent analgesic agent
Shushank Dixit, Pramod Kumar Sharma, Niranjan Kaushik
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 312 KB
Your tags:
english, 2013
41
Microwave-assisted CAN-catalyzed solvent-free synthesis ofN-allyl quinolone-based pyrano[4,3-b]chromene and benzopyrano[3,2-c]chromene derivatives and their antimicrobial activity
Hardik H. Jardosh, Manish P. Patel
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 342 KB
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english, 2013
42
Molecular properties prediction, synthesis, and diuretic activity of phenoxy acetic acid bearing pyrazolines
Mohammed Afroz Bakht, M. Shahar Yar, Anees A. Siddiqui, M. M. Abdullah, Hamadeh Tarazi, Moawiah M. Naffaa, Ahmed M-Alafeefy
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 388 KB
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english, 2013
43
The impact of glycerol and some carbohydrates on antibiotic production byStreptomyces hygroscopicusCH-7
Slavica B. Ilić, Sandra S. Konstantinović, Gordana Đ. Gojgić Cvijović, Dragiša S. Savić, Vlada B. Veljković
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 311 KB
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english, 2013
44
Antibacterial, antifungal and antioxidant activity of some new water-soluble β-diketones
Javed Sheikh, Taibi Ben Hadda
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 772 KB
Your tags:
english, 2013
45
Application of pocket modeling andk-nearest neighbor molecular field analysis (kNN-MFA) for designing of some anticoagulants: potential factor IXa inhibitors
P. B. Choudhari, M. S. Bhatia, N. M. Bhatia
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 596 KB
Your tags:
english, 2013
46
Synthesis and pharmacological evaluation of novel 4-isopropylthiazole-4-phenyl-1,2,4-triazole derivatives as potential antimicrobial and antitubercular agents
G. V. Suresh Kumar, Y. Rajendra Prasad, S. M. Chandrashekar
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 370 KB
Your tags:
english, 2013
47
Synthesis of kojic acid-derived copper-chelating apoptosis inducing agents
Yu-Hua Chen, Pei-Jung Lu, Christopher Hulme, Arthur Y. Shaw
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 514 KB
Your tags:
english, 2013
48
In silicodesigning and characterization of Amiloride derivatives as ion channel modulator
Ajeet
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 571 KB
Your tags:
english, 2013
49
Design, synthesis, anti-inflammatory, analgesic screening, and molecular docking of some novel 2-pyridyl (3H)-quinazolin-4-one derivatives
Ahmad F. Eweas, Ahmed O. H. El-Nezhawy, Ayman R. Baiuomy, Mohamed M. Awad
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 519 KB
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english, 2013
50
Synthesis, characterization, and biological evaluation of certain 1,3-thiazolone derivatives bearing pyrazoline moiety as potential anti-breast cancer agents
Nadia A. Khalil, Eman M. Ahmed, Hala B. El-Nassan
Journal:
Medicinal Chemistry Research
Year:
2013
Language:
english
File:
PDF, 322 KB
Your tags:
english, 2013
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