Volume 23; Issue 12

Medicinal Chemistry Research

Volume 23; Issue 12

1

Quantitative structure–activity relationship (QSAR) studies as strategic approach in drug discovery

Patel, Harun M., Noolvi, Malleshappa N., Sharma, Poonam, Jaiswal, Varun, Bansal, Sumit, Lohan, Sandeep, Kumar, Suthar Sharad, Abbot, Vikrant, Dhiman, Saurabh, Bhardwaj, Varun

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 591 KB

english, 2014

2

Pharmacophore modeling, 3DQSAR, and docking-based design of polysubstituted quinolines derivatives as inhibitors of phosphodiesterase 4, and preliminary evaluation of their anti-asthmatic potential

Gaurav, Anand, Singh, Ranjit

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 6.13 MB

english, 2014

3

Synthesis and antitumor properties of novel alizarin analogs

Yao, Guiyang, Dai, Weilong, Ye, Manyi, Huang, Rizhen, Pan, Ying-ming, Liao, Zhi-Xin, Wang, Heng-shan

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 797 KB

english, 2014

4

Electron affinity and dipole moment of 1,2,4,5-tetraoxanes antimalarials and correlation with activity againstPlasmodium falciparum

de Paula, Mariane C., Valle, Marcelo S., Pliego, Josefredo R.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 461 KB

english, 2014

5

Synthesis and biological evaluation of novel quinolin-2(1H)-one derivatives as potential antimicrobial agents

Deng, Qiao, Ji, Qing-Gang, Ge, Zhi-Qiang, liu, Xiao-Fei, Yang, Dan, Yuan, Lv-Jiang

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 371 KB

english, 2014

6

Synthesis, pharmacophore modeling, and cytotoxic activity of 2-thioxothiazolidin-4-one derivatives

Alegaon, Shankar G., Alagawadi, Kallanagouda R., Vinod, D., Unger, Banappa, Khatib, N. A.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 713 KB

english, 2014

7

Effect of garlic and cabbage on healing of gastric ulcer in experimental rats

Ben Hadda, Taibi, ElSawy, Naser A., Header, Eslam A. M., Mabkhot, Yahia N., Mubarak, Mohammad S.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.20 MB

english, 2014

8

Synthesis of indole-2-hydrazones in search of potential leishmanicidal agents

Taha, Muhammad, Ismail, Nor Hadiani, Ali, Muhammad, Khan, Khalid M., Jamil, Waqas, Kashif, Syed Muhammad, Asraf, Mohammad

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 414 KB

english, 2014

9

In silico molecular docking study of natural compounds on wild and mutated epidermal growth factor receptor

Singh, Pushpendra, Bast, Felix

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 2.31 MB

english, 2014

10

Chemical synthesis, molecular modelling, and evaluation of anticancer activity of some pyrazol-3-one Schiff base derivatives

Bensaber, Salah M., Allafe, H. A., Ermeli, Nouri B., Mohamed, Salah B., Zetrini, Abdulmottaleb A., Alsabri, Sami G., Erhuma, Mabrouk, Hermann, Anton, Jaeda, Mousa I., Gbaj, Abdul M.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.34 MB

english, 2014

11

Synthesis and antibacterial activity of (1-aryl-1, 2, 3-triazol-4-yl) methyl esters of morpholine-3-carboxylic acid

Narsimha, Sirassu, Ranjith Kumar, T., Satheesh Kumar, Nukala, Yakoob, Shaik, Vasudeva Reddy, N.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 999 KB

english, 2014

12

Synthesis, biological evaluation, and molecular docking studies ofN-(α-acetamido cinnamoyl) aryl hydrazone derivatives as antiinflammatory and analgesic agents

Rajitha, Galla, Prasad, Koganti V. S. R. G., Umamaheswari, Amineni, Pradhan, Dibyabhaba, Bharathi, Koganti

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.40 MB

english, 2014

13

Highly potent analgesic activity of monoterpene-derived (2S,4aR,8R,8aR)-2-aryl-4,7-dimethyl-3,4,4a,5,8,8a-hexahydro-2H-chromene-4,8-diols

Il’ina, Irina, Mikhalchenko, Oksana, Pavlova, Alla, Korchagina, Dina, Tolstikova, Tat’yana, Volcho, Konstantin, Salakhutdinov, Nariman, Pokushalov, Evgeniy

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 421 KB

english, 2014

14

Synthesis, biological evaluation of certain pyrazolo[3,4-d]pyrimidines as novel anti-inflammatory and analgesic agents

Kadry, Hanan H.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 700 KB

english, 2014

15

Design, synthesis, crystal structure, bioactivity, and molecular docking studies of novel sulfonylamidine-derived neonicotinoid analogs

Yang, Liu, Zhao, Yong-Long, Zhao, Chun-Yan, Li, Huan-Huan, Wang, Mei-Juan, Morris-Natschke, Susan L., Qian, Keduo, Lee, Kuo-Hsiung, Liu, Ying-Qian

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.92 MB

english, 2014

16

Synthesis and antibacterial activity of novel fluoroquinolone analogs

Dixit, Sandeep Kumar, Yadav, Neesha, Kumar, Satyanand, Good, Liam, Awasthi, Satish K.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.41 MB

english, 2014

17

Insight into the anti-amyloidogenic activity of polyphenols and its application in virtual screening of phytochemical database

Chakraborty, Sandipan, Basu, Soumalee

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 513 KB

english, 2014

18

Molecular modeling of a series of pyridinecarboxamidrazone-azole derivatives with antifungal activity

Terra, Luciana, Castro, Helena Carla, Abreu, Paula Alvarez

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 971 KB

english, 2014

19

Selection of 2D/3D molecular descriptors and QSAR modeling of aromatic Morita–Baylis–Hillman adducts with leishmanicidal activities

Alencar Filho, Edilson B., Weber, Karen C., Vasconcellos, Mário L. A. A.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 483 KB

english, 2014

20

1,3,5-Triazine inhibitors of histone deacetylases: synthesis and biological activity

Zhao, Xiaodong, Tan, Qiu, Zhang, Zhitao, Zhao, Yu

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 986 KB

english, 2014

21

Anticonvulsant effects of bis-1,4-dihydropyridines and the probable role of L-type calcium channels suggested by docking simulations

Ramírez-San Juan, Eduardo, Soriano-Ursúa, Marvin A., Espinosa-Raya, Judith, Correa-Basurto, José, Trujillo-Ferrara, José G., Miranda-Ruvalcaba, René, Delgado-Reyes, Francisco, Gómez-Pliego, Raquel

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.73 MB

english, 2014

22

Synthesis, molecular properties and DFT studies of new phosphoramidates as potential urease inhibitors

Oliveira, Fabricio M., Barbosa, Luiz C. A., Demuner, Antônio J., Maltha, Célia R. A., Pereira, Silvana R., Horta, Lívia P., Modolo, Luzia V.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 527 KB

english, 2014

23

A mild and efficient one-pot three-component synthesis of anti-β-amino-carbonyl compounds catalyzed by NH4OAc and their anticancer activities

Venkatesan, Sathesh, Karthikeyan, Natesan Sundaramoorthy, Rathore, Ravindranath S., Giridharan, Periyasamy, Sathiyanarayanan, Kulathu Iyer

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 828 KB

english, 2014

24

Anti-parkinsonian efficacy of target-specific GSK3β inhibitors demonstrated inCaenorhabditis elegans

Pradeep, H., Shashikumar, S., Rajini, P. S., Rajanikant, G. K.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 911 KB

english, 2014

25

Inhibitors of cytosolic phospholipase A2α with carbamate structure: synthesis, biological activity, metabolic stability, and bioavailability

Schwarzkopf, Julian, Sundermann, Tom, Arnsmann, Martina, Hanekamp, Walburga, Fabian, Jörg, Heidemann, Jan, Pott, Anna Friederike, Bettenworth, Dominik, Lehr, Matthias

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 662 KB

english, 2014

26

Quantitative structure–activity relationship analysis of antibacterial cationic anthraquinone analogs using Hansch and Fujita models

Nziko, V. P. N., Fosso, Marina Y., Chang, Cheng-Wei Tom

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 440 KB

english, 2014

27

Structural requirements for imidazo[1,2-a]pyrazine derivatives as Aurora A kinase inhibitors and validation of the model

Kanhed, Ashish M., Zambre, Vishal P., Pawar, Vijay A., Sharma, Mayank Kumar, Giridhar, Rajani, Yadav, Mange Ram

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 2.45 MB

english, 2014

28

Ritodrine inhibits neuronal nitric oxide synthase, a potential link between tocolysis and autism

Suaifan, Ghadeer A. R. Y., Shehadeh, Mayadah B., Al-Ijel, Hebah A. N., Al-Jamal, Khuloud T., Taha, Mutasem O.

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 519 KB

english, 2014

29

Pentacyclic triterpenoids fromMitracarpus frigidus(Willd. ex Roem. & Schult.) K. Shum: in vitro cytotoxic and leishmanicidal and in vivo anti-inflammatory and antioxidative activities

Fabri, Rodrigo Luiz, Garcia, Roberta Alvim, Florêncio, Jônatas Rodrigues, de Carvalho, Lidiane Oliveira, de Castro Campos Pinto, Nícolas, Coimbra, Elaine Soares, de Souza-Fagundes, Elaine Maria, Ribei

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 430 KB

english, 2014

30

Novel isomannide-based peptide mimetics containing a tartaric acid backbone as serine protease inhibitors

Abrahim-Vieira, Bárbara, da Costa, Emmerson C. B., de A. Azevedo, Pedro H. R., Portela, Aline C., Dias, Luiza R. S., Pinheiro, Sergio, Tanuri, Amilcar, Capaccia, Anne M., Ventura, Gustavo T., Mohana-B

Journal:

Medicinal Chemistry Research

Year:

2014

Language:

english

File:

PDF, 1.05 MB

english, 2014

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