Volume 25; Issue 7

Medicinal Chemistry Research

Volume 25; Issue 7

1

Synthesis, characterization and evaluation of antiproliferative activity of diisopropylphenyl esters of fatty acids from selected oils

Yasa, Sathyam Reddy, Kaki, Shiva Shanker, Rao, Bala Bhaskara, Jain, Nishant, Penumarthy, Vijayalakshmi

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 692 KB

english, 2016

2

Synthesis of new benzimidazole and phenylhydrazinecarbothiomide hybrids and their anticonvulsant activity

Siddiqui, Nadeem, Alam, Md. Shamsher, Ali, Ruhi, Yar, M. Shahar, Alam, Ozair

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 934 KB

english, 2016

3

Design, synthesis and anti-acetylcholinesterase evaluation of some new pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives

Romdhane, Anis, Said, Abderrahim Ben, Cherif, Maher, Jannet, Hichem Ben

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 722 KB

english, 2016

4

In silico molecular docking of niloticin with acetylcholinesterase 1 (AChE1) ofAedes aegyptiL. (Diptera: Culicidae): a promising molecular target

Reegan, Appadurai Daniel, Stalin, Antony, Paulraj, Michael Gabriel, Balakrishna, Kedike, Ignacimuthu, Savarimuthu, Al-Dhabi, Naif Abdullah

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.47 MB

english, 2016

5

Design, synthesis of new chiral fluorine-containing β-hydroxysulfonamides from natural amino acids and study of their anti-inflammatory and analgesic activities

Gloulou, Monia, Kraïem, Jamil, Jennene, Fayçal, Ghedira, Donia, Amor, Haifa Bel Haj, Lajili, Sirine, Jalleli, Emna, Ferjani, Maha, Bouraoui, Abderrahman, Kallel, Mohamed

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 821 KB

english, 2016

6

Formylchromone derivatives as novel and selective PTP-1B inhibitors: a drug design aspect using molecular docking-based self-organizing molecular field analysis

Verma, Sant K., Thareja, Suresh

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 3.59 MB

english, 2016

7

Synthesis and characterization of novel conjugates of 4-[3-(aryl/heteroaryl)-3-oxo-propenyl]-benzaldehyde with thiazole and thiazolidinones as possible voltage-gated sodium channel blockers

Pandey, Sundeep, Sonar, Pankaj K., Saraf, Shailendra K.

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.00 MB

english, 2016

8

Discovery of highly potent analgesic activity of isopulegol-derived (2R,4aR,7R,8aR)-4,7-dimethyl-2-(thiophen-2-yl)octahydro-2H-chromen-4-ol

Nazimova, Ekaterina, Pavlova, Alla, Mikhalchenko, Oksana, Il’ina, Irina, Korchagina, Dina, Tolstikova, Tat’yana, Volcho, Konstantin, Salakhutdinov, Nariman

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 883 KB

english, 2016

9

Binding mode of conformations and structure-based pharmacophore development for farnesyltransferase inhibitors

Moorthy, N. S. Hari Narayana, Sousa, Sergio F., Ramos, Maria J., Fernandes, Pedro A.

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 9.17 MB

english, 2016

10

QSAR studies for some thiazolidine-2,4-dione derivatives as PIM-2 kinase inhibitors

Asati, Vivek, Bharti, Sanjay K.

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.67 MB

english, 2016

11

Synthesis and potential anticonvulsant activity of new aryl sulfonyl semicarbazide derivatives

Nie, Yousong, Zhong, Min, Jiang, Zhiyuan, Sun, Jian, Gao, Yangguang, Ding, Fei, Li, Hang, Zhang, Yongmin, He, Xianran

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 505 KB

english, 2016

12

Design, synthesis, and evaluation of the anticonvulsant and antidepressant activities of pyrido[2,3-d]pyrimidine derivatives

Zhang, Hong-Jian, Wang, Shi-Ben, Wen, Xiang, Li, Jin-Zi, Quan, Zhe-Shan

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 571 KB

english, 2016

13

Synthesis, in vitro and in silico anti-proliferative activity of 4-aryl-4H-chromene derivatives

Parthiban, A., Kumaravel, M., Muthukumaran, J., Rukkumani, R., Krishna, R., Rao, H. Surya Prakash

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 800 KB

english, 2016

14

Piroxicam sulfonates biology-oriented drug synthesis (BIODS), characterization and anti-nociceptive screening

Ullah, Safi, Saeed, Muhammad, Halimi, Syed Muhammad Ashhad, Fakhri, Muhammad Imran, Khan, Khalid Mohammed, Khan, Ikhtiar, Perveen, Shahnaz

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 598 KB

english, 2016

15

HQSAR and molecular docking studies of furanyl derivatives as adenosine A2Areceptor antagonists

Muñoz-Gutiérrez, Camila, Caballero, Julio, Morales-Bayuelo, Alejandro

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.29 MB

english, 2016

16

Synthesis and anticonvulsant activities of functionalized 5-(isoindole-1,3-dione)-pyrimidinones

Sharma, Rashmi, Gawande, Dinesh Y., Mohan, Chander, Goel, Rajesh Kumar

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 483 KB

english, 2016

17

A facile synthesis and neuroprotective role of novel quinoxaline-2,3-bis hydrazones in ethidium bromide-induced demyelinated rats

Rajamanickam, Gayathri, Selvaraj, Jubie, Selvaraj, Suresh, Rajendran, Thirumurthy

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.32 MB

english, 2016

18

Inhibitory effect of 4,4′-[ethane-1,2-diylbis(sulfandiylmethanediyl)]bis(3,5-dimethyl-1H-pyrazole) and its derivatives on alpha-amylase activity

Maksimov, Vadim, Zaynullin, Radik, Akhmadiev, Nail, Segura-Ceniceros, Elda P., Martínez Hernández, José L., Bikbulatova, Elmira, Akhmetova, Vnira, Kunakova, Raijana, Ramos, Rodolfo, Ilyina, Anna

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 658 KB

english, 2016

19

Design, synthesis and evaluation of acridin-9-yl hydrazide derivatives as BACE-1 inhibitors

Jain, Priti, Wadhwa, Pankaj K., Jadhav, Hemant R.

Journal:

Medicinal Chemistry Research

Year:

2016

Language:

english

File:

PDF, 1.32 MB

english, 2016