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Volume 39; Issue 10
Main
Neurochemical Research
Volume 39; Issue 10
Neurochemical Research
Volume 39; Issue 10
1
Probing for Improved Potency and In Vivo Bioavailability of Excitatory Amino Acid Transporter Subtype 1 Inhibitors UCPH-101 and UCPH-102: Design, Synthesis and Pharmacological Evaluation of Substituted 7-Biphenyl Analogs
Erichsen, Mette N.
,
Hansen, Jeanette
,
Ruiz, Josep A.
,
Demmer, Charles S.
,
Abrahamsen, Bjarke
,
Bastlund, Jesper F.
,
Bundgaard, Christoffer
,
Jensen, Anders A.
,
Bunch, Lennart
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 404 KB
Your tags:
english, 2014
2
Inhibition of AMPA Receptors by Polyamine Toxins is Regulated by Agonist Efficacy and Stargazin
Poulsen, Mette H.
,
Lucas, Simon
,
Strømgaard, Kristian
,
Kristensen, Anders S.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 606 KB
Your tags:
english, 2014
3
GABA Pharmacology: The Search for Analgesics
McCarson, Kenneth E.
,
Enna, S. J.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 752 KB
Your tags:
english, 2014
4
Correlating the Metabolic Stability of Psychedelic 5-HT2AAgonists with Anecdotal Reports of Human Oral Bioavailability
Leth-Petersen, Sebastian
,
Bundgaard, Christoffer
,
Hansen, Martin
,
Carnerup, Martin A.
,
Kehler, Jan
,
Kristensen, Jesper Langgaard
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 610 KB
Your tags:
english, 2014
5
mGluR5: Exploration of Orthosteric and Allosteric Ligand Binding Pockets and Their Applications to Drug Discovery
Mølck, Christina
,
Harpsøe, Kasper
,
Gloriam, David E.
,
Mathiesen, Jesper M.
,
Nielsen, Søren M.
,
Bräuner-Osborne, Hans
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 2.09 MB
Your tags:
english, 2014
6
Multi-target Design Strategies in the Context of Alzheimer’s Disease: Acetylcholinesterase Inhibition and NMDA Receptor Antagonism as the Driving Forces
Rosini, Michela
,
Simoni, Elena
,
Minarini, Anna
,
Melchiorre, Carlo
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 833 KB
Your tags:
english, 2014
7
Muscimol as an Ionotropic GABA Receptor Agonist
Johnston, Graham A. R.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 204 KB
Your tags:
english, 2014
8
The GABA Synapse as a Target for Antiepileptic Drugs: A Historical Overview Focused on GABA Transporters
Schousboe, Arne
,
Madsen, Karsten K.
,
Barker-Haliski, Melissa L.
,
White, H. Steve
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 298 KB
Your tags:
english, 2014
9
On the Discovery and Development of Pimavanserin: A Novel Drug Candidate for Parkinson’s Psychosis
Hacksell, Uli
,
Burstein, Ethan S.
,
McFarland, Krista
,
Mills, Roger G.
,
Williams, Hilde
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 1.01 MB
Your tags:
english, 2014
10
Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization
Jørgensen, Lars
,
Nielsen, Birgitte
,
Pickering, Darryl S.
,
Kristensen, Anders S.
,
Frydenvang, Karla
,
Madsen, Ulf
,
Clausen, Rasmus P.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 745 KB
Your tags:
english, 2014
11
Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)
Al-Khawaja, Anas
,
Petersen, Jette G.
,
Damgaard, Maria
,
Jensen, Mette H.
,
Vogensen, Stine B.
,
Lie, Maria E. K.
,
Kragholm, Bolette
,
Bräuner-Osborne, Hans
,
Clausen, Rasmus P.
,
Frølund, Bente
,
Wellendorph
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 446 KB
Your tags:
english, 2014
12
Analysis of γ-Aminobutyric Acid (GABA) Type A Receptor Subtypes Using Isosteric and Allosteric Ligands
Olsen, Richard W.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 688 KB
Your tags:
english, 2014
13
The Receptor Concept in 3D: From Hypothesis and Metaphor to GPCR–Ligand Structures
Kooistra, Albert J.
,
de Graaf, Chris
,
Timmerman, Henk
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 3.19 MB
Your tags:
english, 2014
14
Revision of the Classical Dopamine D2Agonist Pharmacophore Based on an Integrated Medicinal Chemistry, Homology Modelling and Computational Docking Approach
Krogsgaard-Larsen, N.
,
Harpsøe, K.
,
Kehler, J.
,
Christoffersen, C. T.
,
Brøsen, P.
,
Balle, T.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 1.18 MB
Your tags:
english, 2014
15
Group III Metabotropic Glutamate Receptors: Pharmacology, Physiology and Therapeutic Potential
Mercier, Marion S.
,
Lodge, David
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 601 KB
Your tags:
english, 2014
16
Introduction to Special Issue in Honor of Professor Povl Krogsgaard-Larsen
Bräuner-Osborne, Hans
,
Schousboe, Arne
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 179 KB
Your tags:
english, 2014
17
Povl Krogsgaard-Larsen: A Giant in Medicinal Chemistry Research
Bøgesø, Klaus P.
Journal:
Neurochemical Research
Year:
2014
Language:
english
File:
PDF, 108 KB
Your tags:
english, 2014
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