Organic & Biomolecular Chemistry

1

Triple molecular target approach to selective melanoma cytotoxicity

Skibo, Edward B., Jamil, Akmal, Austin, Brittany, Hansen, Douglas, Ghodousi, Armand

Journal:

Year:

2010

Language:

english

File:

PDF, 499 KB

english, 2010

2

N-Heterocycle construction via cyclic sulfamidates. Applications in synthesis

Bower, John F., Rujirawanich, Janjira, Gallagher, Timothy

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 1.39 MB

english, 2010

3

Synthesis of novel 2,5-diarylselenophenes from selenation of 1,4-diarylbutane-1,4-diones or methanol/arylacetylenes

Hua, Guoxiong, Henry, John B., Li, Yang, Mount, Andrew R., Slawin, Alexandra M. Z., Woollins, J. Derek

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 270 KB

english, 2010

4

Complex interactions of pillar[5]arene with paraquats and bis(pyridinium) derivatives

Li, Chunju, Xu, Qianqian, Li, Jian, Feina Yao,, Jia, Xueshun

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 551 KB

english, 2010

5

Nucleophilic attack of 2-sulfinyl acrylates: A mild and general approach to sulfenic acid anions

Singh, Suneel P., O'Donnell, Jennifer S., Schwan, Adrian L.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 189 KB

english, 2010

6

UVA-induced cyclobutane pyrimidine dimers in DNA: a direct photochemical mechanism?

Mouret, Stéphane, Philippe, Coralie, Gracia-Chantegrel, Jocelyne, Banyasz, Akos, Karpati, Szilvia, Markovitsi, Dimitra, Douki, Thierry

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 260 KB

english, 2010

7

Microwave-induced electrostatic etching: generation of highly reactive magnesium for application in Grignard reagent formation

van de Kruijs, Bastiaan H. P., Dressen, Mark H. C. L., Meuldijk, Jan, Vekemans, Jef A. J. M., Hulshof, Lumbertus A.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 332 KB

english, 2010

8

The effects of tryptophan and hydrophobicity on the structure and bioactivity of novel indolicidin derivatives with promising pharmaceutical potential

Podorieszach, Aaron P., Huttunen-Hennelly, Heidi E. K.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 460 KB

english, 2010

9

The thiocarbonyl ‘S’ is softer than thiolate ‘S’: A catalyst-free one-pot synthesis of isothiocyanates in water

Jamir, Latonglila, Ali, Abdur Rezzak, Ghosh, Harisadhan, Chipem, Francis A. S., Patel, Bhisma K.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 189 KB

english, 2010

10

Use of unnatural β-peptides as a self-assembling component in functional organic fibres

Torres, Elisabeth, Puigmartí-Luis, Josep, Pérez del Pino, Ángel, Ortuño, Rosa M., Amabilino, David B.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 418 KB

english, 2010

11

Structurally-variable, rigid and optically-active D2 and D3 macrocycles possessing recognition properties towards C60

Coluccini, Carmine, Dondi, Daniele, Caricato, Marco, Taglietti, Angelo, Boiocchi, Massimo, Pasini, Dario

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 698 KB

english, 2010

12

Preparation of novel alkylated arginine derivatives suitable for click-cycloaddition chemistry and their incorporation into pseudosubstrate- and bisubstrate-based kinase inhibitors

van Ameijde, Jeroen, Poot, Alex J., van Wandelen, Loek T. M., Wammes, Angelique E. M., Ruijtenbeek, Rob, Rijkers, Dirk T. S., Liskamp, Rob M. J.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 436 KB

english, 2010

13

Unexpected transalkylation on 3-alkyl-2-alkylthio-1,3,4-thiadiazolium-5-thiolates: A computational and experimental mechanistic study

Espinosa, Arturo, García, Rafaela, Molina, Pedro, Tárraga, Alberto

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 326 KB

english, 2010

14

Unravelling the stereoselectivity in 6-exo-trig radical cyclization of α,β-unsaturated ester-tethered sugars. A tale of two stereocenters

de Oliveira, Marcelo T., Cesar, Amary, Leal, Daniel H. S., Prado, Maria A. F., da Silva, Thais H. Á., Alves, Ricardo J.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 257 KB

english, 2010

15

The UDP-Galp mutase catalyzed isomerization: synthesis and evaluation of 1,4-anhydro-β-d-galactopyranose and its [2.2.2] methylene homologue

Sadeghi-Khomami, Ali, Forcada, Tatiana J., Wilson, Claire, Sanders, David A. R., Thomas, Neil R.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 254 KB

english, 2010

16

The continuous flow synthesis of butane-2,3-diacetal protected building blocks using microreactors

Carter, Catherine F., Baxendale, Ian R., Pavey, John B. J., Ley, Steven V.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 491 KB

english, 2010

17

Cell adhesion through clustered ligand on fluid supported lipid bilayers

Sandrin, Ludivine, Coche-Guérente, Liliane, Bernstein, Amandine, Basit, Hajra, Labbé, Pierre, Dumy, Pascal, Boturyn, Didier

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 217 KB

english, 2010

18

Design and synthesis of new amino-modified iminocyclitols: selective inhibitors of α-galactosidase

Ganesan, Muthupandian, Madhukarrao, Rekhawar V., Ramesh, Namakkal G.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 146 KB

english, 2010

19

Photoreversible DNA end capping for the formation of hairpin structures

Yoshimura, Yoshinaga, Okada, Hajime, Fujimoto, Kenzo

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 148 KB

english, 2010

20

Fluorescence quenched quinone methide based activity probes – a cautionary tale

Sellars, Jonathan D., Landrum, Marie, Congreve, Aileen, Dixon, David P., Mosely, Jackie A., Beeby, Andrew, Edwards, Robert, Steel, Patrick G.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 560 KB

english, 2010

21

Cyclization kinetics and biological evaluation of an anticancer 1,2-dialkynylimidazole

Laroche, Christophe, Li, Jing, Gonzales, Cristina, David, Wendi M., Kerwin, Sean M.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 320 KB

english, 2010

22

Rhodium-catalyzed [2+2+2] cycloaddition of various fluorine-containing alkynes—novel synthesis of multi-substituted fluoroalkylated aromatic compounds

Konno, Tsutomu, Moriyasu, Kazuki, Kinugawa, Ryoko, Ishihara, Takashi

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 262 KB

english, 2010

23

Design and synthesis of a tetradentate ‘3-amine-1-carboxylate’ ligand to mimic the metal binding environment at the non-heme iron(ii) oxidase active site

Dungan, Victoria J., Ortin, Yannick, Mueller-Bunz, Helge, Rutledge, Peter J.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 405 KB

english, 2010

24

Back cover

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 551 KB

english, 2010

25

Inside front cover

Journal:

Organic & Biomolecular Chemistry

Year:

2010

File:

PDF, 255 KB

2010

26

Formation of 5′,8-cyclo-2′-deoxyadenosine in single strand DNA. Theoretical quantum mechanics study

Karwowski, Boleslaw T.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 310 KB

english, 2010

27

Front cover

Journal:

Organic & Biomolecular Chemistry

Year:

2010

File:

PDF, 250 KB

2010

28

Asymmetric Si–O coupling of alcohols

Weickgenannt, Andreas, Mewald, Marius, Oestreich, Martin

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 738 KB

english, 2010

29

Biosynthesis of the mitochondrial adenine nucleotide translocase (ATPase) inhibitor bongkrekic acid in Burkholderia gladioli

Rohm, Barbara, Scherlach, Kirstin, Hertweck, Christian

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 155 KB

english, 2010

30

Asymmetric total synthesis of 1-deoxy-7,8-di-epi-castanospermine

Zambrano, Vincenzo, Rassu, Gloria, Roggio, Annamaria, Pinna, Luigi, Zanardi, Franca, Curti, Claudio, Casiraghi, Giovanni, Battistini, Lucia

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 229 KB

english, 2010

31

Highly efficient and stereoselective biosynthesis of (2S,5S)-hexanediol with a dehydrogenase from Saccharomyces cerevisiae

Müller, Marion, Katzberg, Michael, Bertau, Martin, Hummel, Werner

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 659 KB

english, 2010

32

Searching for intermediates in Prins cyclisations: the 2-oxa-5-adamantyl carbocation

Alder, Roger W., Carta, Fabrizio, Reed, Christopher A., Stoyanova, Irina, Willis, Christine L.

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 346 KB

english, 2010

33

Fate of monoterpenes in near-critical water and supercritical alcohols assisted by microwave irradiation

Szuppa, Tony, Stolle, Achim, Ondruschka, Bernd

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 289 KB

english, 2010

34

A highly selective ratiometric fluorescent probe for 1,4-dithiothreitol (DTT) detection

Zhu, Baocun, Zhang, Xiaoling, Jia, Hongying, Li, Yamin, Liu, Haipeng, Tan, Weihong

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 274 KB

english, 2010

35

On new N-heterocyclic carbene derived alkylidene imidazolines

Knappke, Christiane E. I., Neudörfl, Jörg M., von Wangelin, Axel Jacobi

Journal:

Organic & Biomolecular Chemistry

Year:

2010

Language:

english

File:

PDF, 439 KB

english, 2010

Volume 8; Issue 7

Triple molecular target approach to selective melanoma cytotoxicity

N-Heterocycle construction via cyclic sulfamidates. Applications in synthesis

Synthesis of novel 2,5-diarylselenophenes from selenation of 1,4-diarylbutane-1,4-diones or methanol/arylacetylenes

Complex interactions of pillar[5]arene with paraquats and bis(pyridinium) derivatives

Nucleophilic attack of 2-sulfinyl acrylates: A mild and general approach to sulfenic acid anions

UVA-induced cyclobutane pyrimidine dimers in DNA: a direct photochemical mechanism?

Microwave-induced electrostatic etching: generation of highly reactive magnesium for application in Grignard reagent formation

The effects of tryptophan and hydrophobicity on the structure and bioactivity of novel indolicidin derivatives with promising pharmaceutical potential

The thiocarbonyl ‘S’ is softer than thiolate ‘S’: A catalyst-free one-pot synthesis of isothiocyanates in water

Use of unnatural β-peptides as a self-assembling component in functional organic fibres

Structurally-variable, rigid and optically-active D2 and D3 macrocycles possessing recognition properties towards C60

Preparation of novel alkylated arginine derivatives suitable for click-cycloaddition chemistry and their incorporation into pseudosubstrate- and bisubstrate-based kinase inhibitors

Unexpected transalkylation on 3-alkyl-2-alkylthio-1,3,4-thiadiazolium-5-thiolates: A computational and experimental mechanistic study

Unravelling the stereoselectivity in 6-exo-trig radical cyclization of α,β-unsaturated ester-tethered sugars. A tale of two stereocenters

The UDP-Galp mutase catalyzed isomerization: synthesis and evaluation of 1,4-anhydro-β-d-galactopyranose and its [2.2.2] methylene homologue

The continuous flow synthesis of butane-2,3-diacetal protected building blocks using microreactors

Cell adhesion through clustered ligand on fluid supported lipid bilayers

Design and synthesis of new amino-modified iminocyclitols: selective inhibitors of α-galactosidase

Photoreversible DNA end capping for the formation of hairpin structures

Fluorescence quenched quinone methide based activity probes – a cautionary tale

Cyclization kinetics and biological evaluation of an anticancer 1,2-dialkynylimidazole

Rhodium-catalyzed [2+2+2] cycloaddition of various fluorine-containing alkynes—novel synthesis of multi-substituted fluoroalkylated aromatic compounds

Design and synthesis of a tetradentate ‘3-amine-1-carboxylate’ ligand to mimic the metal binding environment at the non-heme iron(ii) oxidase active site

Back cover

Inside front cover

Formation of 5′,8-cyclo-2′-deoxyadenosine in single strand DNA. Theoretical quantum mechanics study

Front cover

Asymmetric Si–O coupling of alcohols

Biosynthesis of the mitochondrial adenine nucleotide translocase (ATPase) inhibitor bongkrekic acid in Burkholderia gladioli

Asymmetric total synthesis of 1-deoxy-7,8-di-epi-castanospermine

Highly efficient and stereoselective biosynthesis of (2S,5S)-hexanediol with a dehydrogenase from Saccharomyces cerevisiae

Searching for intermediates in Prins cyclisations: the 2-oxa-5-adamantyl carbocation

Fate of monoterpenes in near-critical water and supercritical alcohols assisted by microwave irradiation

A highly selective ratiometric fluorescent probe for 1,4-dithiothreitol (DTT) detection

Contents

On new N-heterocyclic carbene derived alkylidene imidazolines