Volume 4; Issue 6

Organic Process Research & Development

Volume 4; Issue 6

1

Chemical Development of MDL 103371: An N-Methyl-d-Aspartate-Type Glycine Receptor Antagonist for the Treatment of Stroke†

Watson, Timothy J. N., Horgan, Stephen W., Shah, Ramnik S., Farr, Robert A., Schnettler, Richard A., Nevill, C. Richard, Weiberth, Franz J., Huber, Edward W., Baron, Bruce M., Webster, Mark E.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 166 KB

english, 2000

2

New Economical, Convenient Procedures for the Synthesis of Catecholborane †

Kanth, Josyula V. B., Periasamy, Mariappan, Brown, Herbert C.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 85 KB

english, 2000

3

A Practical Synthesis of Enantiomerically Pure N -Benzyl-α-methyl Benzylamine

Huckabee, Brian K., Lin, Sechoing, Smith, Traci L., Stuk, Timothy L.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 55 KB

english, 2000

4

A Practical Synthesis of an Anti-Methicillin Resistant Staphylococcus aureus Cephalosporin BMS-247243

Singh, Janak, Kim, Oak K., Kissick, Thomas P., Natalie, Kenneth J., Zhang, Bo, Crispino, Gerard A., Springer, Dane M., Wichtowski, John A., Zhang, Yunhui, Goodrich, Jason, Ueda, Yasutsugu, Luh, Bing Y

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 396 KB

english, 2000

5

Convenient Preparation of Functionalised Polymer-Based Resins via an Economical Preparation of Chloromethylated Polystyrene Resins (Merrifield Type)

Carre, Erica Le, Lewis, Norman, Ribas, Christina, Wells, Andrew

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 54 KB

english, 2000

6

A Scaleable Route to the Pure Enantiomers of Verapamil

Bannister, Robin M., Brookes, Michael H., Evans, Graham R., Katz, Ruth B., Tyrrell, Nicholas D.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 196 KB

english, 2000

7

Phosphorus Oxychloride and Acetone: An Incompatibility Investigation Using ARC

Brenek, Steven J., am Ende, David J., Clifford, Pamela J.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 35 KB

english, 2000

8

Practical and Large-Scale Synthesis of r ac -(3 S ,4a R ,10a R )- 6-Methoxy-1-propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[ g ]quinoline-3-carboxylic Acid Methyl Ester

Bänziger, Markus, Cercus, Jacques, Stampfer, Wolfgang, Sunay, Ustun

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 124 KB

english, 2000

9

Application of the Schöpf Method to Optimization of the Synthesis of 3-[2-( p - N -Acetylaminophenyl)ethyl]-3-hydroxy-4-methylpentanoic Acid: Simultaneous Reduction of Three Functional Groups to Maximize Yield and Throughput

Deering, Carl F., Huckabee, Brian K., Lin, Sechoing, Porter, Ken T., Rossman, Craig A., Wemple, James

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 89 KB

english, 2000

10

Automated Process Research. An Example of Accelerated Optimization of the Friedel−Crafts Acylation Reaction, a Key Step for the Synthesis of Anti-HIV (+)-Calanolide A

Zhang, Jintao, Kirchhoff, Eric W., Zembower, David E., Jimenez, Nancy, Sen, Prabir, Xu, Ze-Qi, Flavin, Michael T.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 131 KB

english, 2000

11

High Selectivity in the Oxidation of Mandelic Acid Derivatives and in O- Methylation of Protocatechualdehyde: New Processes for Synthesis of Vanillin, i so- Vanillin, and Heliotropin

Bjørsvik, Hans-René, Liguori, Lucia, Minisci, Francesco

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 295 KB

english, 2000

12

Modulation of Catalyst Reactivity for the Chemoselective Hydrogenation of a Functionalized Nitroarene: Preparation of a Key Intermediate in the Synthesis of ( R , R )-Formoterol Tartrate

Wilkinson, H. Scott, Hett, Robert, Tanoury, Gerald J., Senanayake, Chris H., Wald, Stephen A.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 76 KB

english, 2000

13

Identification and Comparison of Impurities in Fluoxetine Hydrochloride Synthesized by Seven Different Routes

Wirth, David D., Miller, Marybeth S., Boini, Sathish K., Koenig, Thomas M.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 147 KB

english, 2000

14

A Review of U.S. Patents in the Field of Organic Process Development Published during April to July, 2000

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 240 KB

english, 2000

15

Aerobic Oxidation of Methylpyridines to Pyridinecarboxylic Acids Catalyzed by N -Hydroxyphthalimide

Shibamoto, Akihiro, Sakaguchi, Satoshi, Ishii, Yasutaka

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 80 KB

english, 2000

16

Homogeneous RuCl 2 (PPh 3 ) 3 -Catalyzed Regioselective Liquid-Phase Transfer Hydrogenation of Carbon−Carbon Double Bond in Chlorobenzylidene Ketones with Ethylene Glycol as Hydrogen Donor

Mukhopadhyay, Sudip, Yaghmur, Anan, Benichou, Axel, Sasson, Yoel

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 104 KB

english, 2000

17

Process Development of the Sharpless Catalytic Asymmetric Dihydroxylation Reaction To Prepare Methyl (2 R ,3 S )-2,3-Dihydroxy-3-phenylpropionate

Lu, Xinbo, Xu, Zhunle, Yang, Guojun

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 33 KB

english, 2000

18

A Safe and Efficient Process for the Synthesis of the Inhalation Anesthetic Sevoflurane

Ramakrishna, Kornpati, Behme, Chris, Schure, Ralph M., Bieniarz, Christopher

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 42 KB

english, 2000

19

Some Items of Interest to Process R&D Chemists and Engineers as Selected by Trevor Laird and Stephen A. Hermitage

Hermitage, Stephen A.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 162 KB

english, 2000

20

Large-Scale Synthesis of a Key Catalytic Reagent for Phosphorus Protection in Building Blocks for Isopolar Phosphonate Oligonucleotide Preparation

Rejman, Dominik, Erbs, Jiří, Rosenberg, Ivan

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 65 KB

english, 2000

21

Factors Affecting the Selectivity of Air Oxidation Of 2-Ethyhexanal, an α-Branched Aliphatic Aldehyde

Lehtinen, Christel, Brunow, Gösta

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 86 KB

english, 2000

22

10.1021/op000104u

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 18 KB

english, 2000

23

Development of a New Synthetic Route of a Non-Peptide CCR5 Antagonist, TAK-779, for Large-Scale Preparation

Ikemoto, Tomomi, Ito, Tatsuya, Hashimoto, Hideo, Kawarasaki, Tadao, Nishiguchi, Atsuko, Mitsudera, Hiroyuki, Wakimasu, Mitsuhiro, Tomimatsu, Kiminori

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 66 KB

english, 2000

24

The Use of PeptiCLEC-TR in the Preparation of Dipeptides

Faulconbridge, Susan J., Holt, Karen E., Lock, Christopher J., Taylor, Stephen J. C., Woods, Martin

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 45 KB

english, 2000

25

Development and Scale Up of a Route to Cyclohexylhydrazine Dimethanesulfonate

Connolly, Terrence J., Crittall, Andrew J., Ebrahim, Alkarim S., Ji, Guijun

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 43 KB

english, 2000

26

Application of Focused Microwaves to the Scale-Up of Solvent-Free Organic Reactions

Cléophax, J., Liagre, M., Loupy, A., Petit, A.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 408 KB

english, 2000

27

Rapid Process Development and Scale-Up Using A Multiple Reactor System

Simms, Cormac, Singh, Jasbir

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 161 KB

english, 2000

28

A Facile, One-Pot Procedure for the Preparation of 2-Phenyl-1,3-propanediol Monocarbamate, a Metabolite of Felbamate

Miller, Thomas A., Dieckhaus, Christine M., Macdonald, Timothy L.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 25 KB

english, 2000

29

From Adenosine to 3‘-Deoxyadenosine: Development and Scale Up

Aman, Sayed, Anderson, D. Jason, Connolly, Terrence J., Crittall, Andrew J., Ji, Guijun

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 53 KB

english, 2000

30

Racemisation of R -Bupivacaine: A Key Factor in the Integrated and Economic Process for the Production of Levobupivacaine

Langston, Marianne, Dyer, Ulrich C., Frampton, Graham A. C., Hutton, Gordon, Lock, Christopher J., Skead, Benjamin M., Woods, Martin, Zavareh, Hooshang S.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 41 KB

english, 2000

31

Kinetics and Process Parameter Studies in Oxidative Chlorination of 4-Methylphenol under Phase-Transfer Conditions

Mukhopadhyay, Sudip, Mukhopadhyaya, Jayanta K., Ponde, Datta E., Cohen, Shlomo, Kurkalli, Basan G. S.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 79 KB

english, 2000

32

Efficient Molar-Scale Synthesis of 1-Methyl-5-acylimidazole Triflic Acid Salts

Chen, Bang-Chi, Skoumbourdis, Amanda P., Sundeen, Joseph E., Rovnyak, George C., Traeger, Sarah C.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 28 KB

english, 2000

33

On-Line Monitoring of Vacuum Dryers Using Mass Spectrometry

am Ende, David J., Preigh, Michael J., Hettenbach, Kevin, Ahlijanian, Paul, Ward, Howard W.

Journal:

Organic Process Research & Development

Year:

2000

Language:

english

File:

PDF, 88 KB

english, 2000

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