Volume 9; Issue 1

Organic Process Research & Development

Volume 9; Issue 1

1

Synthesis of Commercial Phosphodiesterase(V) Inhibitors

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 430 KB

english, 2005

2

DioRaSSP: Diosynth Rapid Solution Synthesis of Peptides

Bakelaar, Frits T., Petersen, Annet, Ten Kortenaar, Paul B. W., Eggen, Ivo F.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 203 KB

english, 2005

3

An Expeditious Scalable Synthesis of ( S )-2-Amino-5-methoxytetralin via Resolution

Hirayama, Yoshihiro, Ikunaka, Masaya, Matsumoto, Jun

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 222 KB

english, 2005

4

Viral Clearance Issues Associated with the Use of an Animal-Derived Enzyme in the Synthesis of Emtricitabine

Gaede, Bruce J., Nardelli, Christy A.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 92 KB

english, 2005

5

Efficient and Scalable Method for the Selective Alkylation and Acylation of Secondary Amines in the Presence of Primary Amines

Laduron, Frédéric, Tamborowski, Vanessa, Moens, Luc, Horváth, András, De Smaele, Dirk, Leurs, Stef

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 51 KB

english, 2005

6

Investigation of Practical Routes for the Kilogram-Scale Production of cis -3-Methylamino-4-methylpiperidines

Cai, Weiling, Colony, James L., Frost, Heather, Hudspeth, James P., Kendall, Peter M., Krishnan, Ashwin M., Makowski, Teresa, Mazur, Duane J., Phillips, James, Ripin, David H. Brown, Ruggeri, Sally Gu

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 149 KB

english, 2005

7

Aza-Diels−Alder Reaction of Methyl 2-[( R )-1-Phenylethyl]iminoethanoate with Cyclopentadiene Using Practical and Environmentally Friendly Biphasic Solvent System

Hashimoto, Norio, Yasuda, Hironobu, Hayashi, Masaru, Tanabe, Yoo

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 67 KB

english, 2005

8

A Facile and Scaleable Synthesis of ABT-239, A Benzofuranoid H 3 Antagonist

Pu, Yu-Ming, Grieme, Timothy, Gupta, Ashok, Plata, Daniel, Bhatia, Ashok V., Cowart, Marlon, Ku, Yi-Yin

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 81 KB

english, 2005

9

Process Development and Scale-up of a Selective α 1 -Adrenoceptor Antagonist

Connolly, Terrence J., Matchett, Michael, Sarma, Keshab

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 118 KB

english, 2005

10

Some Items of Interest to Process R&D Chemists and Engineers

Laird, Trevor, Hermitage, Stephen A., Tilstam, Ulf

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 189 KB

english, 2005

11

Minimizing Isobutylene Emissions from Large Scale tert -Butoxycarbonyl Deprotections

Dias, Eric L., Hettenbach, Kevin W., am Ende, David J.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 102 KB

english, 2005

12

Polymeric Materials in Organic Synthesis and Catalysis Edited by Michael R. Buchmeiser. Wiley Interscience: Weinheim. 2003. xxxiii + 559 pp. 159 Euro/235 SFR. ISBN 3-527-30630-7.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 20 KB

english, 2005

13

A Review of U.S. Patents in the Field of Organic Process Development Published during September and October 2004

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 168 KB

english, 2005

14

Chemical Micro Process Engineering: Fundamentals, Modelling and Reactions, 10th ed by V. Hessel, S. Hardt, and H. Löwe. Kluwer Academic Publishers: Dordrecht. 2003. Wiley-VCH: Weinheim. 2004. xxxviii + 674 pp. £135. ISBN 3-527-30741-9.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 20 KB

english, 2005

15

The Chemistry of Process Development in Fine Chemical & Pharmaceutical Industry By C. Someswara Rao. Asian Books Private Limited: New Delhi. 2004. 1277 pp. ISBN 81-86299-50-5.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 7 KB

english, 2005

16

Does Industry Get Its Synthetic Methodology on the Cheap?

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 17 KB

english, 2005

17

Practical Process for the Air Oxidation of Cresols: Part B. Evaluation of the Laboratory-Scale Oxidation Process

Barton, Benita, Logie, Catherine G., Schoonees, Barbara M., Zeelie, Bernard

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 145 KB

english, 2005

18

Practical Process for the Air Oxidation of Cresols: Part A. Mechanistic Investigations

Barton, Benita, Logie, Catherine G., Schoonees, Barbara M., Zeelie, Bernard

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 129 KB

english, 2005

19

Practical Synthesis of Triethylammonium ( Z )-2-[2-(Boc-amino)thiazol-4-yl]-2-(trityloxyimino)acetate, the Side Chain of Cefmatilen

Goto, Yoshihisa, Masui, Yoshiyuki, Kitaura, Yoji, Kobayashi, Tatsuya, Takahashi, Hisanori, Okuyama, Akira

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 78 KB

english, 2005

20

Optimisation of Ethyl(2-phthalimidoethoxy)acetate Synthesis with the Aid of DOE

Synoradzki, Ludwik, Jańczewski, Dominik, Włostowski, Marek

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 342 KB

english, 2005

21

A Study of the Paterson Boron Aldol Reaction as Used in the Large-Scale Total Synthesis of the Anticancer Marine Natural Product (+)-Discodermolide

Mickel, Stuart J., Daeffler, Robert, Prikoszovich, Walter

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 156 KB

english, 2005

22

An Efficient Catalytic Asymmetric Route to 1-Aryl-2-imidazol-1-yl-ethanols

Lennon, Ian C., Ramsden, James A.

Journal:

Organic Process Research & Development

Year:

2005

Language:

english

File:

PDF, 62 KB

english, 2005